SCHEMBL19976947

SCHEMBL19976947

CC(NC(=O)c1cccs1)C(=O)Nc1cccc2c1CCCC2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 7/20 0.53
KMT2A Q03164 7/20 0.53
L3MBTL1 Q9Y468 4/20 0.48
KDM4E B2RXH2 2/20 0.48
ALDH1A1 P00352 7/20 0.47
LMNA P02545 5/20 0.46
THRB P10828 2/20 0.46
THRA P10827 1/20 0.46
HPGD P15428 5/20 0.45
HSD17B10 Q99714 4/20 0.45
SMN1; SMN2 Q16637 4/20 0.45
MAPK1 P28482 3/20 0.45
CASP1 P29466 3/20 0.45
CASP7 P55210 3/20 0.45
TSHR P16473 3/20 0.45
NPC1 O15118 3/20 0.45
RAB9A P51151 2/20 0.45
ESR1 P03372 1/20 0.45
TP53 P04637 1/20 0.45
ALOX15 P16050 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18261131 0.82 HSPA1A (0.57) MEN1KMT2AL3MBTL1KDM4EALDH1A1
SCHEMBL16999833 0.82 HSPA1A (0.57) MEN1KMT2AL3MBTL1KDM4EALDH1A1
SCHEMBL19976897 0.81 L3MBTL1 (0.55) MEN1KMT2AL3MBTL1KDM4EALDH1A1
SCHEMBL19976901 0.80 GAA (0.59) MEN1KMT2AL3MBTL1ALDH1A1LMNA
SCHEMBL19977089 0.79 L3MBTL1 (0.52) MEN1KMT2AL3MBTL1KDM4EALDH1A1
SCHEMBL12308333 0.76 ALDH1A1 (0.62) MEN1KMT2AL3MBTL1KDM4EALDH1A1
SCHEMBL19977040 0.76 MAPT (0.71) MEN1KMT2AKDM4EALDH1A1LMNA
SCHEMBL19976914 0.76 PARP1 (0.54) MEN1KMT2AMAPK1NPC1RAB9A
SCHEMBL19976988 0.75 MEN1 (0.52) MEN1KMT2AL3MBTL1KDM4EALDH1A1
SCHEMBL19977042 0.75 KMT2A (0.52) MEN1KMT2AL3MBTL1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3102193-B1 ANTIBACTERIAL AGENTS: N(ALPHA)-AROYL-N-ARYL-PHENYLALANINAMIDES UNIV RUTGERS (US) 2023-01-11 EP disclosed
US-9919998-B2 Antibacterial agents: Nα-aroyl-N-aryl-phenylalaninamides RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2018-03-20 US disclosed