SCHEMBL19984007

SCHEMBL19984007

CNCc1cn(Sc2cccnc2)c2cc(Nc3ccc(OC(F)(F)F)cc3F)ccc12

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAT2A P31153 1/20 0.34
ABL1 P00519 6/20 0.33
BCR P11274 3/20 0.33
KDR P35968 1/20 0.33
KIT P10721 2/20 0.33
DHODH Q02127 1/20 0.33
TRPA1 O75762 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
ROCK2 O75116 1/20 0.31
P2RX7 Q99572 2/20 0.31
SYK P43405 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19983844 0.91 ALDH1A1 (0.35) KITCYP11B1CYP11B2
SCHEMBL19984203 0.91 ABL1 (0.35) MAT2AABL1BCRKDRKIT
SCHEMBL19983777 0.86 ADRB2 (0.37) TRPA1NPC1RAB9AP2RX7
SCHEMBL19984127 0.86 NUDT1 (0.36) MAT2AKDRCYP11B1CYP11B2CYP2C9
SCHEMBL19983721 0.86 HTR2C (0.32) ROCK2
SCHEMBL19983812 0.85 CYP11B1 (0.38) MAT2AABL1BCRCYP11B1CYP11B2
SCHEMBL19984009 0.85 ALPL (0.37) KDRCYP3A4CYP2C9CYP2C19
SCHEMBL19983981 0.84 CNR2 (0.34) KDRCYP3A4CYP2C9CYP2C19
SCHEMBL19983879 0.83
SCHEMBL19983874 0.82 CYP19A1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP disclosed