SCHEMBL19984050

SCHEMBL19984050

CCNCc1c[nH]c2cc(Nc3ccc(OC)nc3Cl)ccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.42
CYP2C8 P10632 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP3A4 P08684 1/20 0.42
KCNH2 Q12809 1/20 0.42
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CACNA1G O43497 1/20 0.36
CACNA1B Q00975 1/20 0.36
HTR2A P28223 2/20 0.35
BCHE P06276 2/20 0.33
ACHE P22303 2/20 0.33
ADORA2A P29274 1/20 0.33
ULK1 O75385 1/20 0.33
PRKAG1 P54619 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16626544 0.90 GPR84 (0.36) CYP2C9MEN1KMT2AKDM4EALDH1A1
SCHEMBL19984013 0.79 HTR2A (0.35) CYP2C19CYP2C9CYP3A4MEN1KMT2A
SCHEMBL19983894 0.76 GPR84 (0.39) CYP1A2CYP2C8CYP2D6CYP2C19CYP2C9
SCHEMBL19983834 0.75 PRKAG1 (0.42) MEN1KMT2ASMN1; SMN2ACHEPRKAG1
SCHEMBL19983877 0.73 GPR84 (0.36) MEN1KMT2AKDM4EALDH1A1SMN1; SMN2
SCHEMBL19983764 0.72 APP (0.38) CYP1A2CYP2C8CYP2D6CYP2C19CYP2C9
SCHEMBL19983880 0.72 MEN1 (0.36) MEN1KMT2AKDM4EALDH1A1SMN1; SMN2
SCHEMBL19983815 0.70 CYP2C9 (0.43) CYP2C19CYP2C9CYP3A4MEN1KMT2A
SCHEMBL19984194 0.70 GPR84 (0.39) CYP1A2CYP2C8CYP2D6CYP2C19KDM4E
SCHEMBL19984147 0.68 CYP2D6 (0.36) CYP1A2CYP2C8CYP2D6CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP disclosed