SCHEMBL20002255

SCHEMBL20002255

CC(=O)N1CCC(C(=O)N2CCC(Sc3ccc(F)cc3)C2)CC1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.49
RORC P51449 5/20 0.45
TACR1 P25103 5/20 0.44
TACR2 P21452 3/20 0.44
KMT2A Q03164 1/20 0.44
NR1I2 O75469 1/20 0.44
TACR3 P29371 4/20 0.43
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
ACACB O00763 1/20 0.42
ACACA Q13085 1/20 0.42
HSD11B1 P28845 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002719 0.87 HSD11B1 (0.48) KMT2AHSD11B1
SCHEMBL20003196 0.87 HSD11B1 (0.48) KMT2AHSD11B1
SCHEMBL20002936 0.86 CCR5 (0.46) CCR5TACR1KMT2ATACR3HDAC3
SCHEMBL20002886 0.82 KMT2A (0.40) CCR5RORCKMT2AHSD11B1
SCHEMBL20002972 0.80 L3MBTL1 (0.41) RORCKMT2AHSD11B1
SCHEMBL20002297 0.79 NOTUM (0.47) CCR5RORCKMT2AHSD11B1
SCHEMBL20002430 0.78 RORC (0.44) CCR5RORCKMT2ANR1I2HDAC3
SCHEMBL20002879 0.77 NPC1 (0.44) CCR5KMT2A
SCHEMBL20003220 0.76 RORC (0.41) CCR5RORCKMT2AHSD11B1
SCHEMBL20003024 0.76 NOTUM (0.44) CCR5KMT2AHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed