SCHEMBL20002719

SCHEMBL20002719

O=C(C1CCCCC1)N1CCC(Sc2ccc(F)cc2)C1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.45
ALDH1A1 P00352 3/20 0.43
KMT2A Q03164 2/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
TSHR P16473 1/20 0.42
EPHX2 P34913 1/20 0.41
POLB P06746 1/20 0.41
MEN1 O00255 1/20 0.41
PTPN1 P18031 1/20 0.40
TP53 P04637 1/20 0.40
KEAP1 Q14145 1/20 0.40
PRKAB2 O43741 1/20 0.40
PRKAG1 P54619 1/20 0.40
PRKAA2 P54646 1/20 0.40
PRKAA1 Q13131 1/20 0.40
PRKAG3 Q9UGI9 1/20 0.40
PRKAG2 Q9UGJ0 1/20 0.40
PRKAB1 Q9Y478 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20003196 1.00 HSD11B1 (0.48) HSD11B1L3MBTL1ALDH1A1KMT2AMAPK1
SCHEMBL20002255 0.87 CCR5 (0.49) HSD11B1KMT2A
SCHEMBL20003224 0.87 KMT2A (0.43) HSD11B1ALDH1A1KMT2ASMN1; SMN2TSHR
SCHEMBL20002972 0.87 L3MBTL1 (0.41) HSD11B1L3MBTL1KMT2A
SCHEMBL20003223 0.84 KMT2A (0.41) HSD11B1ALDH1A1KMT2ATSHRMEN1
SCHEMBL20003024 0.81 NOTUM (0.44) HSD11B1L3MBTL1ALDH1A1KMT2AEPHX2
SCHEMBL20002886 0.79 KMT2A (0.40) HSD11B1ALDH1A1KMT2ASMN1; SMN2TP53
SCHEMBL20002297 0.78 NOTUM (0.47) HSD11B1L3MBTL1KMT2A
SCHEMBL4107783 0.77 ALDH1A1 (0.42) ALDH1A1KMT2ASMN1; SMN2POLB
SCHEMBL5472049 0.77 HSD11B1 (0.62) HSD11B1ALDH1A1KMT2APOLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed