SCHEMBL20003091

SCHEMBL20003091

O=C(c1cccc2cnccc12)N1CCC(S(=O)(=O)c2ccc(F)cc2)C1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.54
P2RX7 Q99572 4/20 0.42
GRM4 Q14833 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
NPC1 O15118 1/20 0.41
NR2F2 P24468 1/20 0.41
ROCK2 O75116 1/20 0.39
CCR2 P41597 1/20 0.39
ROCK1 Q13464 1/20 0.39
CHRM1 P11229 1/20 0.39
NAMPT P43490 3/20 0.39
HCRTR1 O43613 2/20 0.39
HCRTR2 O43614 2/20 0.39
NAAA Q02083 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002502 0.80 L3MBTL1 (0.64) ALDH1A1LMNAL3MBTL1NAMPTRAB9A
SCHEMBL23951553 0.77 ALDH1A1 (0.50) ALDH1A1LMNANPC1NR2F2NAMPT
SCHEMBL27478359 0.77 ALDH1A1 (0.50) RORCP2RX7ALDH1A1LMNANPC1
SCHEMBL30098408 0.74 CCR5 (0.53) ALDH1A1LMNANPC1HCRTR1HCRTR2
SCHEMBL23924217 0.74 CCR5 (0.53) ALDH1A1LMNANPC1HCRTR1HCRTR2
SCHEMBL20003002 0.73 TSHR (0.48) RORCALDH1A1L3MBTL1NAMPTRAB9A
SCHEMBL20002837 0.72 RORC (0.49) RORCALDH1A1NAMPT
SCHEMBL14413535 0.71 EPHX2 (0.47) RORCL3MBTL1
SCHEMBL20003085 0.71 PROKR1 (0.44) L3MBTL1NPC1NAMPTRAB9A
SCHEMBL16886748 0.71 RORC (1.00) RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed