SCHEMBL20002890

SCHEMBL20002890

NC(=O)c1ccc(CC(=O)N2CC[C@H]([S+]([O-])c3ccc(F)cc3)C2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.48
ALDH1A1 P00352 2/20 0.48
PARP10 Q53GL7 1/20 0.42
RORC P51449 1/20 0.42
POLB P06746 2/20 0.42
KDM1A O60341 1/20 0.40
KMT2A Q03164 3/20 0.40
PKM P14618 2/20 0.40
LMNA P02545 1/20 0.39
F2 P00734 1/20 0.39
PRSS1 P07477 1/20 0.39
TPSAB1 Q15661 1/20 0.39
TPSD1 Q9BZJ3 1/20 0.39
TPSG1 Q9NRR2 1/20 0.39
ME2 P23368 1/20 0.39
ME1 P48163 1/20 0.39
ME3 Q16798 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MLNR O43193 1/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002912 0.90 ALDH1A1 (0.52) SMN1; SMN2ALDH1A1POLBKDM1AKMT2A
SCHEMBL20002218 0.85 SMN1; SMN2 (0.47) SMN1; SMN2ALDH1A1RORCPOLBPKM
SCHEMBL20002209 0.85 SMN1; SMN2 (0.47) SMN1; SMN2ALDH1A1RORCPOLBPKM
SCHEMBL20003082 0.82 SMN1; SMN2 (0.44) SMN1; SMN2ALDH1A1RORCPOLBPKM
SCHEMBL20003187 0.80 RORC (0.43) SMN1; SMN2ALDH1A1RORCPOLBPKM
SCHEMBL19702977 0.76 SMN1; SMN2 (0.53) SMN1; SMN2ALDH1A1POLBKMT2AL3MBTL1
SCHEMBL20002918 0.75 PKM (0.47) SMN1; SMN2ALDH1A1RORCPOLBKMT2A
SCHEMBL20002495 0.74 RORC (0.40) SMN1; SMN2ALDH1A1RORCKMT2APKM
SCHEMBL20002981 0.73 KDM4E (0.55) SMN1; SMN2ALDH1A1POLBKMT2ALMNA
SCHEMBL20002870 0.73 PDK2 (0.38) SMN1; SMN2ALDH1A1RORCKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed