SCHEMBL20003082

SCHEMBL20003082

O=C(Cc1cncnc1)N1CCC([S+]([O-])c2ccc(F)cc2)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.44
ALDH1A1 P00352 2/20 0.44
RORC P51449 2/20 0.41
PKM P14618 2/20 0.39
MAPT P10636 1/20 0.39
ALOX12 P18054 1/20 0.39
CYP19A1 P11511 1/20 0.38
POLB P06746 2/20 0.38
CYP3A4 P08684 3/20 0.36
IDO1 P14902 2/20 0.36
LMNA P02545 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
TACR3 P29371 1/20 0.36
CNR1 P21554 1/20 0.36
CYP2D6 P10635 1/20 0.35
CYP2B6 P20813 1/20 0.35
MLNR O43193 1/20 0.35
ME2 P23368 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002209 0.88 SMN1; SMN2 (0.47) SMN1; SMN2ALDH1A1RORCPKMMAPT
SCHEMBL20002218 0.88 SMN1; SMN2 (0.47) SMN1; SMN2ALDH1A1RORCPKMMAPT
SCHEMBL20003187 0.85 RORC (0.43) SMN1; SMN2ALDH1A1RORCPKMMAPT
SCHEMBL20002912 0.83 ALDH1A1 (0.52) SMN1; SMN2ALDH1A1PKMMAPTALOX12
SCHEMBL20002890 0.82 SMN1; SMN2 (0.48) SMN1; SMN2ALDH1A1RORCPKMMAPT
SCHEMBL20002918 0.78 PKM (0.47) SMN1; SMN2ALDH1A1RORCPKMPOLB
SCHEMBL20002495 0.77 RORC (0.40) SMN1; SMN2ALDH1A1RORCPKMMAPT
SCHEMBL20002981 0.76 KDM4E (0.55) SMN1; SMN2ALDH1A1POLBLMNA
SCHEMBL20002400 0.75 TACR3 (0.42) SMN1; SMN2ALDH1A1RORCMAPTTACR3
SCHEMBL20002698 0.75 HSD11B1 (0.47) SMN1; SMN2ALDH1A1RORCPOLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed