SCHEMBL20003130

SCHEMBL20003130

O=C(Cc1ccncc1)N1CCC(Sc2ccc(F)cc2)C1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CYP19A1 P11511 1/20 0.44
POLB P06746 3/20 0.42
RORC P51449 5/20 0.42
KDM4E B2RXH2 2/20 0.42
GAA P10253 1/20 0.42
PKM P14618 2/20 0.41
MAPT P10636 1/20 0.41
ALOX12 P18054 1/20 0.41
TACR3 P29371 1/20 0.41
FNTA P49354 1/20 0.40
FNTB P49356 1/20 0.40
USP2 O75604 1/20 0.40
LMNA P02545 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002762 0.88 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2CYP19A1POLBRORC
SCHEMBL20002747 0.82 MAPT (0.44) ALDH1A1SMN1; SMN2CYP19A1POLBRORC
SCHEMBL20003072 0.80 RORC (0.43) ALDH1A1SMN1; SMN2CYP19A1RORCPKM
SCHEMBL20002837 0.76 RORC (0.49) ALDH1A1SMN1; SMN2CYP19A1RORCKDM4E
SCHEMBL20002218 0.75 SMN1; SMN2 (0.47) ALDH1A1SMN1; SMN2CYP19A1POLBRORC
SCHEMBL20002209 0.75 SMN1; SMN2 (0.47) ALDH1A1SMN1; SMN2CYP19A1POLBRORC
SCHEMBL19702601 0.74 MAPT (0.55) ALDH1A1SMN1; SMN2POLBGAAMAPT
SCHEMBL19703195 0.73 SMN1; SMN2 (0.52) ALDH1A1SMN1; SMN2POLBGAAMAPT
SCHEMBL4703997 0.73 FNTA (0.53) ALDH1A1SMN1; SMN2CYP19A1POLBKDM4E
SCHEMBL20002719 0.72 HSD11B1 (0.48) ALDH1A1SMN1; SMN2POLBTSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed