SCHEMBL20002762

SCHEMBL20002762

O=C(Cc1ccnnc1)N1CCC(Sc2ccc(F)cc2)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
RORC P51449 3/20 0.42
PKM P14618 2/20 0.39
MAPT P10636 1/20 0.39
ALOX12 P18054 1/20 0.39
CYP19A1 P11511 1/20 0.38
POLB P06746 2/20 0.38
TP53 P04637 1/20 0.37
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
TACR3 P29371 1/20 0.36
USP2 O75604 1/20 0.36
KCNH2 Q12809 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
KMT2A Q03164 1/20 0.36
CNR1 P21554 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20003130 0.88 ALDH1A1 (0.49) ALDH1A1SMN1; SMN2RORCPKMMAPT
SCHEMBL20002747 0.80 MAPT (0.44) ALDH1A1SMN1; SMN2RORCMAPTCYP19A1
SCHEMBL20003072 0.77 RORC (0.43) ALDH1A1SMN1; SMN2RORCPKMMAPT
SCHEMBL20003187 0.77 RORC (0.43) ALDH1A1SMN1; SMN2RORCPKMMAPT
SCHEMBL20003196 0.72 HSD11B1 (0.48) ALDH1A1SMN1; SMN2POLBTP53TSHR
SCHEMBL20002719 0.72 HSD11B1 (0.48) ALDH1A1SMN1; SMN2POLBTP53TSHR
SCHEMBL19702601 0.72 MAPT (0.55) ALDH1A1SMN1; SMN2MAPTPOLBKMT2A
SCHEMBL19703195 0.71 SMN1; SMN2 (0.52) ALDH1A1SMN1; SMN2MAPTPOLBKMT2A
SCHEMBL20002255 0.70 CCR5 (0.49) RORCTACR3KMT2A
SCHEMBL20002879 0.69 NPC1 (0.44) ALDH1A1SMN1; SMN2LMNAMAPK1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed