SCHEMBL20003152

SCHEMBL20003152

O=C(O)C1(C(=O)N2CCC(Sc3ccc(F)cc3)C2)CC[S+]([O-])CC1

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.34
NPC1 O15118 1/20 0.34
ATM Q13315 1/20 0.34
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
CCR5 P51681 1/20 0.32
ALDH1A1 P00352 2/20 0.32
PKM P14618 1/20 0.32
KMT2A Q03164 1/20 0.31
RBP4 P02753 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CACNA1B Q00975 2/20 0.31
HSD11B1 P28845 6/20 0.31
NOTUM Q6P988 1/20 0.30
DDB1 Q16531 1/20 0.30
CRBN Q96SW2 1/20 0.30
EGFR P00533 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20003154 0.80 RORC (0.39) RAB9ANPC1ATMGRIN1GRIN2B
SCHEMBL20003191 0.78 RORC (0.41) RAB9ANPC1ATMGRIN1GRIN2B
SCHEMBL20002430 0.74 RORC (0.44) CCR5KMT2A
SCHEMBL20002823 0.74 CCR5 (0.38) RAB9ANPC1ATMGRIN1GRIN2B
SCHEMBL20003080 0.73 GRIN1 (0.35) RAB9ANPC1ATMGRIN1GRIN2B
SCHEMBL20002375 0.73 RORC (0.41) RAB9ANPC1ATMGRIN1GRIN2B
SCHEMBL20002612 0.73 RORC (0.36) RAB9ANPC1ATMGRIN1GRIN2B
SCHEMBL20003220 0.73 RORC (0.41) RAB9ANPC1ATMGRIN1GRIN2B
SCHEMBL20003026 0.72 RORC (0.47) RAB9ANPC1ATMGRIN1GRIN2B
SCHEMBL20003131 0.72 RORC (0.46) RAB9ANPC1GRIN1GRIN2BCCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed