SCHEMBL20003026

SCHEMBL20003026

O=C(O)C1CCC(CF)(C(=O)N2CC[C@H](Sc3ccc(F)cc3)C2)CC1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RORC P51449 10/20 0.47
NOTUM Q6P988 1/20 0.38
MAPT P10636 2/20 0.36
CCR5 P51681 1/20 0.35
KMT2A Q03164 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
RAB9A P51151 2/20 0.34
NPC1 O15118 1/20 0.34
ATM Q13315 1/20 0.34
HSD11B1 P28845 1/20 0.34
NR1I2 O75469 1/20 0.33
CACNA1B Q00975 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002297 0.79 NOTUM (0.47) RORCNOTUMMAPTCCR5KMT2A
SCHEMBL20003154 0.78 RORC (0.39) RORCNOTUMMAPTCCR5KMT2A
SCHEMBL20003024 0.77 NOTUM (0.44) NOTUMMAPTCCR5KMT2AGRIN1
SCHEMBL20003191 0.76 RORC (0.41) RORCNOTUMMAPTCCR5KMT2A
SCHEMBL20002823 0.74 CCR5 (0.38) MAPTCCR5KMT2AGRIN1GRIN2B
SCHEMBL20003080 0.73 GRIN1 (0.35) RORCMAPTCCR5KMT2AGRIN1
SCHEMBL20002972 0.73 L3MBTL1 (0.41) RORCNOTUMMAPTKMT2AGRIN1
SCHEMBL20002375 0.73 RORC (0.41) RORCCCR5KMT2AGRIN1GRIN2B
SCHEMBL20003220 0.73 RORC (0.41) RORCMAPTCCR5KMT2AGRIN1
SCHEMBL20003152 0.72 RAB9A (0.34) NOTUMMAPTCCR5KMT2AGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed