SCHEMBL20003131

SCHEMBL20003131

CNC(=O)C1(C(=O)N2CCC(Sc3ccc(F)cc3)C2)CCS(=O)(=O)CC1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RORC P51449 6/20 0.46
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34
CCR5 P51681 1/20 0.33
FAAH O00519 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
KMT2A Q03164 1/20 0.32
EPHX2 P34913 2/20 0.32
HSD11B1 P28845 1/20 0.32
GRIN1 Q05586 1/20 0.31
GRIN2B Q13224 1/20 0.31
UBE2M P61081 1/20 0.31
DCUN1D1 Q96GG9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002430 0.74 RORC (0.44) RORCCCR5KMT2A
SCHEMBL20002823 0.74 CCR5 (0.38) NPC1MAPTRAB9ACCR5SMN1; SMN2
SCHEMBL20003154 0.73 RORC (0.39) RORCNPC1MAPTRAB9ACCR5
SCHEMBL20003220 0.72 RORC (0.41) RORCNPC1MAPTRAB9ACCR5
SCHEMBL20003152 0.72 RAB9A (0.34) NPC1MAPTRAB9ACCR5SMN1; SMN2
SCHEMBL20003191 0.71 RORC (0.41) RORCNPC1MAPTRAB9ACCR5
SCHEMBL20003080 0.71 GRIN1 (0.35) RORCNPC1MAPTRAB9ACCR5
SCHEMBL20002375 0.70 RORC (0.41) RORCNPC1RAB9ACCR5FAAH
SCHEMBL20002407 0.70 SMN1; SMN2 (0.41) NPC1RAB9ACCR5FAAHSMN1; SMN2
SCHEMBL20002294 0.69 PTPN11 (0.36) RORCCCR5KMT2AGRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed