SCHEMBL2002225

SCHEMBL2002225

O=C(c1cnc(-c2ccncc2)o1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2)c2ccc(O)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 4/20 0.39
ALOX5 P09917 2/20 0.39
MAPT P10636 3/20 0.36
PKM P14618 3/20 0.36
KDM4E B2RXH2 2/20 0.36
S1PR3 Q99500 2/20 0.35
ESR1 P03372 1/20 0.35
CCR9 P51686 1/20 0.35
PTGES2 Q9H7Z7 2/20 0.34
GAA P10253 2/20 0.34
ALDH1A1 P00352 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
CNR1 P21554 1/20 0.34
ABCB11 O95342 1/20 0.34
LMNA P02545 2/20 0.33
P2RX3 P56373 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2003925 0.94 ALOX5 (0.39) ALOX5APALOX5MAPTKDM4ECCR9
SCHEMBL2005862 0.92 MAPT (0.41) ALOX5APALOX5MAPTPKMKDM4E
SCHEMBL2002564 0.92 L3MBTL1 (0.36) ALOX5APALOX5MAPTPKMKDM4E
SCHEMBL2007478 0.91 PTGES2 (0.42) ALOX5APALOX5MAPTPKMKDM4E
SCHEMBL2010313 0.91 FAAH (0.42) ALOX5APALOX5MAPTKDM4EPTGES2
SCHEMBL2004831 0.89 PTGES2 (0.38) KDM4ES1PR3PTGES2ALDH1A1CNR1
SCHEMBL2005117 0.89 ALOX5AP (0.36) ALOX5APALOX5MAPTPKMKDM4E
SCHEMBL2001177 0.88 ALOX5AP (0.43) ALOX5APALOX5MAPTPKMALDH1A1
SCHEMBL2007363 0.88 ALOX5AP (0.40) ALOX5APALOX5MAPTPKMKDM4E
SCHEMBL1997676 0.88 ALOX5AP (0.45) ALOX5APALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed