SCHEMBL2003477

SCHEMBL2003477

O=C(c1nnc(-c2ccccn2)o1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2Cl)c2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPT P10636 1/20 0.40
ALOX12 P18054 1/20 0.40
NPSR1 Q6W5P4 3/20 0.38
TSHR P16473 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP3A4 P08684 1/20 0.38
PMP22 Q01453 1/20 0.38
HIF1A Q16665 1/20 0.38
KDM4E B2RXH2 1/20 0.37
OPRK1 P41145 4/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP2C19 P33261 1/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004659 0.95 KDM4E (0.37) LMNAALDH1A1MAPTALOX12NPSR1
SCHEMBL2008404 0.92 L3MBTL1 (0.39) LMNAALDH1A1MAPTALOX12NPSR1
SCHEMBL2001936 0.92 OPRK1 (0.36) LMNAALDH1A1MAPTALOX12NPSR1
SCHEMBL2003403 0.91 LMNA (0.38) LMNAALDH1A1MAPTALOX12NPSR1
SCHEMBL2003372 0.90 PLA2G2A (0.38) MAPTCYP1A2CYP2D6CYP2C9CYP3A4
SCHEMBL2002649 0.89 LMNA (0.43) LMNAALDH1A1MAPTALOX12NPSR1
SCHEMBL2005704 0.89 FAAH (0.39) LMNAALDH1A1MAPTCYP1A2CYP2D6
SCHEMBL2004340 0.89 F2RL3 (0.37) LMNAMAPTKDM4EOPRK1FAAH
SCHEMBL2012451 0.88 LMNA (0.42) LMNAALDH1A1MAPTALOX12NPSR1
SCHEMBL2008181 0.88 LMNA (0.42) LMNAALDH1A1MAPTALOX12NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed