SCHEMBL20042743

SCHEMBL20042743

Cc1cc(C(=O)N2Cc3nc(C)nc(N4CCC4)c3C2)cc(C)n1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.40
PROKR1 Q8TCW9 1/20 0.39
CHRM4 P08173 2/20 0.37
CYP1A2 P05177 1/20 0.37
GBA1 P04062 11/20 0.37
HPGD P15428 2/20 0.35
KDM4E B2RXH2 2/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
GPR55 Q9Y2T6 1/20 0.34
TSHR P16473 1/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
HSD17B10 Q99714 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MTOR P42345 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042872 0.89 P2RX7 (0.44) P2RX7PROKR1CHRM4GBA1CNR1
SCHEMBL20042689 0.88 P2RX7 (0.39) P2RX7PROKR1GBA1CNR2CASP1
SCHEMBL20042829 0.88 P2RX7 (0.41) P2RX7GBA1HPGDKDM4ECNR1
SCHEMBL20042839 0.85 P2RX7 (0.45) P2RX7GBA1HPGDKDM4ECNR1
SCHEMBL20042817 0.85 PKM (0.44) P2RX7GBA1HPGDKDM4E
SCHEMBL20042854 0.85 GRM5 (0.42) P2RX7PROKR1GBA1HPGDKDM4E
SCHEMBL20042671 0.85 P2RX7 (0.45) P2RX7GBA1HPGDCNR1CNR2
SCHEMBL20042755 0.84 GRM5 (0.43) P2RX7GBA1HPGDKDM4ETSHR
SCHEMBL20042873 0.84 P2RX7 (0.38) P2RX7GBA1HPGDKDM4ECNR1
SCHEMBL20042668 0.84 HPGD (0.51) P2RX7GBA1HPGDKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed