SCHEMBL20042867

SCHEMBL20042867

CCn1cc(C(=O)N2Cc3nc(C)nc(N4CCC4)c3C2C)cn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PROKR1 Q8TCW9 8/20 0.39
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP11B1 P15538 2/20 0.34
CYP11B2 P19099 1/20 0.34
KDM4E B2RXH2 3/20 0.33
ALDH1A1 P00352 2/20 0.33
PIK3CD O00329 1/20 0.33
NAMPT P43490 1/20 0.33
POLB P06746 1/20 0.33
HPGD P15428 1/20 0.32
GAA P10253 1/20 0.32
TSHR P16473 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C19 P33261 1/20 0.31
GFER P55789 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042857 0.88 PROKR1 (0.35) PROKR1RAB9ACYP11B1KDM4EALDH1A1
SCHEMBL20042742 0.80 PROKR1 (0.35) PROKR1KMT2AKDM4EALDH1A1POLB
SCHEMBL20042844 0.79 P2RX7 (0.33) KMT2AKDM4EPIK3CDSMN1; SMN2MAPT
SCHEMBL20042865 0.79 TACR3 (0.42) CYP2C19
SCHEMBL20042958 0.79 TACR3 (0.42) CYP2C19
SCHEMBL20042982 0.79 P2RX7 (0.46) KMT2AALDH1A1POLBGAASMN1; SMN2
SCHEMBL20042851 0.79 P2RX7 (0.46) KMT2AALDH1A1POLBGAASMN1; SMN2
SCHEMBL20042767 0.78 TACR3 (0.44) ALDH1A1
SCHEMBL20042896 0.77 GRM5 (0.38) LMNA
SCHEMBL20042766 0.77 TACR3 (0.36) KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed