SCHEMBL2005357

SCHEMBL2005357

Cc1ccc2c(c1)c(C(=O)c1ncc(-c3ccccc3)o1)c(Cl)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 1/20 0.38
ALOX12 P18054 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
PMP22 Q01453 1/20 0.38
HIF1A Q16665 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.36
NPC1 O15118 1/20 0.36
HPGD P15428 1/20 0.35
PTGDR2 Q9Y5Y4 4/20 0.35
PTGS1 P23219 1/20 0.35
SLC26A4 O43511 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2002487 0.94 LMNA (0.40) LMNASMN1; SMN2NPSR1ALDH1A1MAPT
SCHEMBL2006660 0.92 CYP2C9 (0.37) LMNASMN1; SMN2ALDH1A1MAPTALOX12
SCHEMBL2000766 0.92 FAAH (0.36) LMNASMN1; SMN2NPSR1ALDH1A1MAPT
SCHEMBL2007718 0.91 L3MBTL1 (0.43) LMNASMN1; SMN2NPSR1ALDH1A1MAPT
SCHEMBL2001701 0.90 MEN1 (0.42) PTGDR2ALOX5APAKR1B1FAAHCES1
SCHEMBL2005400 0.90 PPARG (0.36) LMNASMN1; SMN2NPSR1ALDH1A1MAPT
SCHEMBL2001270 0.89 FAAH (0.41) FAAH
SCHEMBL2006669 0.89 PLA2G2A (0.41) LMNAALDH1A1MAPTCYP1A2CYP3A4
SCHEMBL2003998 0.89 SLC26A4 (0.40) LMNASMN1; SMN2NPSR1ALDH1A1MAPT
SCHEMBL2006262 0.86 CYP2C9 (0.40) LMNANPSR1ALDH1A1MAPTALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed