SCHEMBL2006257

SCHEMBL2006257

O=C(O)Cc1cn(Cc2ccc(O)cc2)c2c(O)cccc12

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.50
LMNA P02545 1/20 0.50
PLA2G2A P14555 1/20 0.45
CA2 P00918 1/20 0.42
CAMK2A Q9UQM7 1/20 0.42
PPARD Q03181 4/20 0.41
PPARG P37231 3/20 0.41
PPARA Q07869 3/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNA7 P36544 1/20 0.41
CHRNA4 P43681 1/20 0.41
AKR1B1 P15121 1/20 0.41
ABCB1 P08183 2/20 0.41
DNTT P04053 1/20 0.40
HRH1 P35367 1/20 0.40
CDC25A P30304 1/20 0.39
CHRM1 P11229 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MCL1 Q07820 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1997691 0.92 ALDH1A1 (0.58) ALDH1A1LMNAPLA2G2APPARDPPARG
SCHEMBL2004279 0.87 LMNA (0.54) ALDH1A1LMNAPLA2G2APPARDPPARG
SCHEMBL2003339 0.87 LMNA (0.48) ALDH1A1LMNAPLA2G2ACA2CAMK2A
SCHEMBL2008295 0.84 AKR1B1 (0.56) ALDH1A1LMNAAKR1B1ABCB1CDC25A
SCHEMBL2007475 0.79 ALDH1A1 (0.50) ALDH1A1LMNAPLA2G2ACA2CAMK2A
SCHEMBL2002884 0.76 PLA2G2A (0.56) ALDH1A1LMNAPLA2G2ACA2CAMK2A
SCHEMBL2008743 0.76 PLA2G2A (0.70) ALDH1A1LMNAPLA2G2ACA2CAMK2A
SCHEMBL2002819 0.75 LMNA (0.52) ALDH1A1LMNAPLA2G2APPARDPPARG
SCHEMBL2006388 0.74 AKR1B1 (0.50) ALDH1A1LMNACA2AKR1B1ABCB1
SCHEMBL2004958 0.74 PLA2G2A (0.43) PLA2G2ACA2CAMK2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8884020-B2 Indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2014-11-11 US disclosed
US-8884020-B2 Indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2014-11-11 US disclosed
EP-2610244-A1 Indole compounds Ironwood Pharmaceuticals, Inc. (US) 2013-07-03 EP disclosed
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed
US-20100197708-A1 INDOLE COMPOUNDS WELLS FARGO BANK, NATIONAL ASSOCIATION 2010-08-05 US disclosed
US-20100197708-A1 INDOLE COMPOUNDS WELLS FARGO BANK, NATIONAL ASSOCIATION 2010-08-05 US disclosed
US-20090264653-A1 USEFUL INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. 2009-10-22 US disclosed
US-20090264653-A1 USEFUL INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. 2009-10-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100197708-A1 INDOLE COMPOUNDS IDO1, IDO2, TPH2 ALDH1A1 1229/4885LMNA 3450/4885PLA2G2A 3285/4885
US-20090264653-A1 USEFUL INDOLE COMPOUNDS FAAH, FAAH2, AANAT ALDH1A1 178/4885LMNA 4536/4885PLA2G2A 326/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.