SCHEMBL20064061

SCHEMBL20064061

C=CCc1cc(O[C@H]2C[C@H](C(=O)O)C2)c2occc2c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
ENPP2 Q13822 5/20 0.33
CYP3A4 P08684 2/20 0.33
PTGS1 P23219 2/20 0.33
ALDH1A1 P00352 1/20 0.33
ALOX5 P09917 1/20 0.33
AR P10275 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.33
TDP1 Q9NUW8 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
PPARA Q07869 2/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
REN P00797 1/20 0.32
KDM4E B2RXH2 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21222642 0.80 PDE4A (0.39) PDE4APDE4BPDE4CPDE4DENPP2
SCHEMBL21222641 0.80 PDE4A (0.39) PDE4APDE4BPDE4CPDE4DENPP2
SCHEMBL20064596 0.79 MEN1 (0.35) ENPP2ALDH1A1MEN1KMT2ANPC1
SCHEMBL20064291 0.76 LMNA (0.43) CYP3A4MEN1KMT2A
SCHEMBL20064134 0.74 ENPP2 (0.38) PDE4APDE4BPDE4CPDE4DENPP2
SCHEMBL21222645 0.74 ENPP2 (0.38) PDE4APDE4BPDE4CPDE4DENPP2
SCHEMBL20064420 0.74 PPARA (0.57) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL7349242 0.73 ALDH1A1 (0.53) CYP3A4PTGS1ALDH1A1ALOX5AR
SCHEMBL20064062 0.70 PPARA (0.31) PPARAKDM4E
SCHEMBL7351472 0.70 DRD2 (0.34) CYP3A4PTGS1ALDH1A1ALOX5AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018069863-A1 1,3 DI-SUBSTITUTED CYCLOBUTANE OR AZETIDINE DERIVATIVES AS HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-04-19 WO disclosed