SCHEMBL2007964

SCHEMBL2007964

O=C(c1cnc(-c2cccnc2)o1)c1c(Cl)n(Cc2cccc(Cl)c2)c2ccc(O)cc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.41
GRIN2B Q13224 1/20 0.41
HDAC6 Q9UBN7 3/20 0.41
HDAC1 Q13547 2/20 0.41
MAPT P10636 4/20 0.38
ALDH1A1 P00352 3/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
MAPK10 P53779 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
GAA P10253 2/20 0.37
PKM P14618 2/20 0.37
P2RX7 Q99572 1/20 0.37
KDM4E B2RXH2 3/20 0.37
LMNA P02545 3/20 0.37
POLB P06746 1/20 0.37
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2003239 0.93 PTGES2 (0.41) HDAC6HDAC1MAPTALDH1A1CYP1A2
SCHEMBL2004973 0.89 PTGES2 (0.42) GRIN1GRIN2BHDAC6HDAC1MAPT
SCHEMBL2002287 0.89 L3MBTL1 (0.39) HDAC6HDAC1MAPTALDH1A1CYP1A2
SCHEMBL2004791 0.84 MAPT (0.44) MAPTALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL2002956 0.84 PTGES2 (0.44) HDAC6HDAC1MAPTALDH1A1CYP1A2
SCHEMBL2007363 0.83 ALOX5AP (0.40) HDAC6HDAC1MAPTALDH1A1GAA
SCHEMBL1998318 0.83 HDAC6 (0.44) HDAC6HDAC1MAPTALDH1A1CYP1A2
SCHEMBL2003941 0.83 P2RX7 (0.38) HDAC6HDAC1MAPTALDH1A1CYP1A2
SCHEMBL2007478 0.83 PTGES2 (0.42) HDAC6HDAC1MAPTALDH1A1CYP1A2
SCHEMBL2002482 0.82 ALDH1A1 (0.44) MAPTALDH1A1CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed