SCHEMBL2010193

SCHEMBL2010193

CC(C)(C)OC(=O)n1ccc(CN2CCN(C(=O)O)[C@@](C)(Cc3ccccc3)C2)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
POLB P06746 1/20 0.35
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
ACKR3 P25106 1/20 0.33
GPR119 Q8TDV5 1/20 0.33
ACHE P22303 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33
HTR2C P28335 1/20 0.33
SLC6A4 P31645 1/20 0.33
STS P08842 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32
TP53 P04637 2/20 0.32
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2007650 0.76 POLB (0.39) POLBALDH1A1KDM4EGAA
SCHEMBL2010191 0.73 PDK1 (0.50) GPR119SLC6A4HDAC1
SCHEMBL3131491 0.71 MGLL (0.44) GPR119
SCHEMBL1703971 0.71 ALDH1A1 (0.51) POLBALDH1A1KDM4ECHRM2CHRM3
SCHEMBL14813528 0.71 ALDH1A1 (0.45) OPRD1OPRK1NR1H2NR1H3ACHE
SCHEMBL1703908 0.70 ALDH1A1 (0.43) POLBALDH1A1KDM4EHDAC1
SCHEMBL1633895 0.70 KDM4E (0.51) POLBALDH1A1KDM4EMAPT
SCHEMBL12878388 0.70 CYP4F2 (0.43) POLBNR1H2NR1H3MAPTHDAC1
SCHEMBL1188920 0.69 MEN1 (0.48) ALDH1A1KDM4EGAA
SCHEMBL14085918 0.68 NPFFR1 (0.47) OPRD1OPRK1ACHEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7964602-B2 Biaryl compounds useful as agonists of the Gpr38 receptor GLAXO GROUP LIMITED (GB) 2011-06-21 US disclosed