SCHEMBL20109593

SCHEMBL20109593

NCc1cccc(COC(N)=O)c1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.52
LOXL2 Q9Y4K0 3/20 0.49
NOS1 P29475 5/20 0.46
NOS2 P35228 5/20 0.46
NOS3 P29474 3/20 0.46
ALDH1A1 P00352 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
CYP3A4 P08684 1/20 0.46
NFKB1 P19838 1/20 0.46
MRGPRX4 Q96LA9 1/20 0.44
CFD P00746 1/20 0.43
PLG P00747 1/20 0.43
PLAU P00749 1/20 0.43
F11 P03951 1/20 0.43
KLKB1 P03952 1/20 0.43
F7 P08709 1/20 0.43
TPSB2 P20231 1/20 0.43
LMNA P02545 1/20 0.43
PNMT P11086 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9677464 0.92 LMNA (0.48) ALDH1A1LMNA
Benzyl Carbamate SCHEMBL9998168 0.87 ALDH1A1 (0.55) LOXL2ALDH1A1LMNA
SCHEMBL28330985 0.85 PRKCA (0.47) ENPP2NOS1NOS2NOS3ALDH1A1
SCHEMBL5709288 0.84 TPSAB1 (0.51) LOXL2ALDH1A1PLG
SCHEMBL6648255 0.84 ALDH1A1 (0.43) LOXL2ALDH1A1SMN1; SMN2LMNA
Urethane SCHEMBL28735644 0.84 ALOX15 (0.54) ENPP2LOXL2NOS1NOS2NOS3
SCHEMBL27795850 0.84 LMNA (0.42) ALDH1A1LMNA
SCHEMBL29011017 0.84 ENPP2 (0.50) ENPP2LOXL2NOS1NOS2NOS3
SCHEMBL31139242 0.84 ALDH1A1 (0.43) ALDH1A1LMNA
SCHEMBL27664520 0.84 ALDH1A1 (0.61) ENPP2LOXL2NOS1NOS2NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2534152-B1 MACROCYCLES AS FACTOR XIA INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-05-02 EP disclosed