SCHEMBL20118182

SCHEMBL20118182

COC/C1=N/N(c2ccc(F)cc2Cl)C(=O)CCCCC1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.39
MAPK13 O15264 2/20 0.36
MAPK12 P53778 2/20 0.36
MAPK11 Q15759 2/20 0.36
MAPK14 Q16539 2/20 0.36
CASP6 P55212 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36
P2RX7 Q99572 7/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
GRM5 P41594 2/20 0.34
CNR1 P21554 1/20 0.33
OXTR P30559 2/20 0.33
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20118221 0.87 MAPK13 (0.38) PDE4BMAPK13MAPK12MAPK11MAPK14
SCHEMBL20118039 0.81 KMT2A (0.46) MAPK13MAPK12MAPK11MAPK14CASP6
SCHEMBL20118399 0.73 P2RX7 (0.39) MAPK13MAPK12MAPK11MAPK14CASP6
SCHEMBL20103445 0.68 P2RX7 (0.52) CASP6KMT2AMEN1GAAP2RX7
SCHEMBL20118223 0.68 GRM5 (0.33) P2RX7ALDH1A1GRM5OXTR
SCHEMBL20118389 0.68 GRM5 (0.33) P2RX7ALDH1A1GRM5OXTR
SCHEMBL20118222 0.68 OPRL1 (0.34) CASP6KMT2AMEN1GAAP2RX7
SCHEMBL20118049 0.67 CASP6 (0.36) CASP6KMT2AMEN1GAAP2RX7
SCHEMBL20118185 0.67 OPRM1 (0.35) CASP6KMT2AMEN1GAAP2RX7
SCHEMBL20118237 0.65 MEN1 (0.41) CASP6KMT2AMEN1GAAP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018078009-A1 AMIDO-SUBSTITUTED CYCLOHEXANE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-03 WO disclosed