SCHEMBL20118221

SCHEMBL20118221

CC/C1=N/N(c2ccc(F)cc2Cl)C(=O)CCCCC1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK13 O15264 2/20 0.38
MAPK12 P53778 2/20 0.38
MAPK11 Q15759 2/20 0.38
MAPK14 Q16539 2/20 0.38
KMT2A Q03164 3/20 0.38
CASP6 P55212 2/20 0.38
MEN1 O00255 2/20 0.38
GAA P10253 1/20 0.38
P2RX7 Q99572 9/20 0.37
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
SHMT2 P34897 1/20 0.35
ADRA1B P35368 1/20 0.34
PDE4B Q07343 1/20 0.34
PER2 O15055 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20118182 0.87 PDE4B (0.39) MAPK13MAPK12MAPK11MAPK14KMT2A
SCHEMBL20118399 0.85 P2RX7 (0.39) MAPK13MAPK12MAPK11MAPK14KMT2A
SCHEMBL20118039 0.84 KMT2A (0.46) MAPK13MAPK12MAPK11MAPK14KMT2A
SCHEMBL20118185 0.71 OPRM1 (0.35) KMT2ACASP6MEN1GAAP2RX7
SCHEMBL20103445 0.71 P2RX7 (0.52) KMT2ACASP6MEN1GAAP2RX7
SCHEMBL20118237 0.68 MEN1 (0.41) KMT2ACASP6MEN1GAAP2RX7
SCHEMBL20118397 0.68 P2RX7 (0.35) KMT2ACASP6MEN1GAAP2RX7
SCHEMBL20118049 0.67 CASP6 (0.36) KMT2ACASP6MEN1GAAP2RX7
SCHEMBL20118169 0.64 P2RX7 (0.35) P2RX7
SCHEMBL16759677 0.63 ALDH1A1 (0.65) KMT2AMEN1P2RX7ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018078009-A1 AMIDO-SUBSTITUTED CYCLOHEXANE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-03 WO disclosed