SCHEMBL20118288

SCHEMBL20118288

CC/C=C(\CC)C(=O)Nc1ccc(C(=N)NC(=O)OCCCC(=O)OC(C)(C)C)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.36
NPC1 O15118 4/20 0.36
SMN1; SMN2 Q16637 4/20 0.36
HPGD P15428 3/20 0.36
CASP1 P29466 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HDAC8 Q9BY41 1/20 0.34
ALDH1A1 P00352 2/20 0.33
MAPK1 P28482 2/20 0.33
BCL2 P10415 1/20 0.33
BECN1 Q14457 1/20 0.33
RECQL P46063 1/20 0.32
TSHR P16473 1/20 0.32
KDM4E B2RXH2 2/20 0.32
MAPT P10636 2/20 0.32
MCL1 Q07820 1/20 0.32
POLB P06746 1/20 0.32
KMT2A Q03164 1/20 0.32
GLA P06280 1/20 0.32
EPHX2 P34913 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20118347 0.78 MEN1 (0.39) HPGDALDH1A1KDM4EKMT2APTPN11
SCHEMBL20118291 0.78 LMNA (0.40) RAB9ANPC1SMN1; SMN2HDAC8ALDH1A1
SCHEMBL24765305 0.77 L3MBTL1 (0.40) RAB9ANPC1SMN1; SMN2HPGDL3MBTL1
SCHEMBL22382076 0.71 ADRB2 (0.39) RAB9ANPC1ALDH1A1TSHRMAPT
SCHEMBL20118645 0.70 CYP19A1 (0.42) RAB9ANPC1SMN1; SMN2HPGDTSHR
SCHEMBL20118630 0.69 F2 (0.61)
SCHEMBL20118453 0.69 RAB9A (0.47) RAB9ANPC1SMN1; SMN2HPGDCASP1
SCHEMBL4417206 0.66 PPID (0.47) SMN1; SMN2L3MBTL1ALDH1A1TSHRKDM4E
SCHEMBL20118820 0.66 F2 (0.34) RAB9ANPC1SMN1; SMN2HPGDALDH1A1
SCHEMBL27523391 0.64 PRMT1 (0.45) NPC1ALDH1A1MAPTGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081513-A1 PRODRUGS OF KALLIKREIN INHIBITORS BIOCRYST PHARMACEUTICALS, INC. (US) 2018-05-03 WO disclosed