SCHEMBL2012375

SCHEMBL2012375

O=C(c1ncc(-c2ccncn2)o1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2)c2ccc(O)cc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 2/20 0.37
MAPT P10636 4/20 0.34
PKM P14618 3/20 0.34
KDM4E B2RXH2 3/20 0.34
ALOX5AP P20292 3/20 0.34
ALOX5 P09917 2/20 0.34
SCD O00767 2/20 0.33
SCD5 Q86SK9 2/20 0.33
PTGES2 Q9H7Z7 1/20 0.33
CCR9 P51686 1/20 0.33
GAA P10253 2/20 0.32
ALDH1A1 P00352 2/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
ABCB11 O95342 1/20 0.32
S1PR3 Q99500 1/20 0.32
LMNA P02545 1/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2007801 0.94 FAAH (0.38) FAAHMAPTKDM4EALOX5APALOX5
SCHEMBL2006590 0.91 FAAH (0.40) FAAHMAPTKDM4EALOX5APALOX5
SCHEMBL2000665 0.91 L3MBTL1 (0.35) FAAHMAPTSCDSCD5ALDH1A1
SCHEMBL2001846 0.90 FAAH (0.41) FAAH
SCHEMBL2000914 0.90 FAAH (0.42) FAAHMAPTKDM4ESCDSCD5
SCHEMBL2002457 0.90 ALOX5 (0.36) MAPTPKMKDM4EALOX5APALOX5
SCHEMBL2004890 0.89 FAAH (0.39) FAAHMAPTPKMKDM4EALOX5AP
SCHEMBL2008885 0.89 LMNA (0.41) FAAHMAPTPKMKDM4EALOX5AP
SCHEMBL2009198 0.89 ALOX5AP (0.39) FAAHMAPTPKMALOX5APALOX5
SCHEMBL2004892 0.87 LMNA (0.35) FAAHMAPTPKMKDM4EALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed