SCHEMBL20140363

SCHEMBL20140363

CC1(c2ccc(F)cc2)CCN(c2ccc(-c3ccccc3)c(F)c2F)C1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.34
HTR7 P34969 1/20 0.34
KIT P10721 1/20 0.33
EPHX2 P34913 1/20 0.33
HSD11B1 P28845 2/20 0.32
RORC P51449 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
OPRL1 P41146 1/20 0.32
NPY1R P25929 1/20 0.32
HTR1A P08908 1/20 0.31
DRD2 P14416 1/20 0.31
DRD3 P35462 1/20 0.31
CYP3A4 P08684 2/20 0.31
USP2 O75604 1/20 0.31
TSHR P16473 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20140426 0.72 HTR6 (0.43) HTR7HTR1A
SCHEMBL20140471 0.65 RORC (0.37) CYP2D6HSD11B1RORCCYP3A4HDAC1
SCHEMBL24685649 0.64 SIGMAR1 (0.46) OPRM1DRD2MEN1KMT2A
SCHEMBL10533047 0.62 ALOX5AP (0.53) DRD3TSHRHDAC2CYP2C9CYP2C19
SCHEMBL6926354 0.62 OPRM1 (0.51) CYP2D6OPRM1OPRD1DRD2KMT2A
SCHEMBL9230998 0.61 MAOB (0.43) HSD11B1
SCHEMBL27099783 0.59 OPRM1 (0.63) EPHX2OPRM1OPRD1OPRK1
SCHEMBL24119449 0.59 OPRM1 (0.63) EPHX2OPRM1OPRD1OPRK1
SCHEMBL8931777 0.59 OPRM1 (0.63) EPHX2OPRM1OPRD1OPRK1
SCHEMBL10819384 0.59 HSD11B1 (0.51) HSD11B1OPRM1OPRD1OPRK1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538522-A1 ROR GAMMA MODULATORS Bristol-Myers Squibb Company (US) 2019-09-18 EP disclosed
WO-2018089406-A1 ROR GAMMA MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed