SCHEMBL20140943

SCHEMBL20140943

CC(C)(C)C1CN(C(=O)O)Cc2nc(-c3ccccc3)nn21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 7/20 0.40
ADORA1 P30542 6/20 0.40
DPP4 P27487 1/20 0.40
DPP8 Q6V1X1 1/20 0.40
DPP7 Q9UHL4 1/20 0.40
NR1H2 P55055 2/20 0.37
NR1H3 Q13133 2/20 0.37
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35
TSHR P16473 1/20 0.35
F2 P00734 1/20 0.34
CYP1A2 P05177 1/20 0.34
MAPT P10636 1/20 0.34
CYP2C9 P11712 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.34
GAA P10253 1/20 0.34
PDK2 Q15119 2/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20141429 0.72 DPP4 (0.54) ADORA3ADORA1DPP4DPP8DPP7
SCHEMBL20140942 0.68 CKS1B (0.49) ADORA3ADORA1DPP4DPP8DPP7
SCHEMBL3393288 0.59 NR1H2 (0.63) ADORA1NR1H2NR1H3RAB9ANPC1
SCHEMBL13677263 0.59 HRH4 (0.47) ADORA3ADORA1DPP4DPP8DPP7
SCHEMBL16003887 0.58 PDE10A (0.45) NR1H2NR1H3TSHRKMT2AALDH1A1
SCHEMBL3118565 0.57 MTHFD2 (0.50) TSHR
SCHEMBL4959931 0.57 DRD2 (0.62) RAB9AHPGDKMT2A
SCHEMBL8650872 0.57 GAA (0.57) ADORA1NR1H2NR1H3TSHRF2
SCHEMBL28739860 0.56 P2RX7 (0.55) ALDH1A1LMNA
SCHEMBL1696532 0.56 LMNA (0.54) TSHRMAPTHPGDKMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed