SCHEMBL21362523

SCHEMBL21362523

C=Cc1ccc(C(=O)c2ccc(CS(=O)(=O)N(C)C(=O)OC(C)(C)C)cc2Br)cc1OC

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACHE P22303 7/20 0.33
LSS P48449 2/20 0.33
BCHE P06276 4/20 0.32
ALDH1A1 P00352 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
PTPN1 P18031 3/20 0.31
MTNR1A P48039 2/20 0.31
MTNR1B P49286 2/20 0.31
PDF Q9HBH1 1/20 0.30
HTT P42858 1/20 0.30
AAK1 Q2M2I8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157726 0.88 ACHE (0.34) ACHEBCHEALDH1A1MTNR1AMTNR1B
SCHEMBL20158056 0.88 ACHE (0.35) ACHEBCHEALDH1A1MTNR1AMTNR1B
SCHEMBL21362533 0.78 ACHE (0.43) ACHELSSBCHEALDH1A1PTPN1
SCHEMBL21564703 0.74 MAPT (0.33) ALDH1A1NPSR1HTT
SCHEMBL21550462 0.73 NPC1 (0.36) ALDH1A1
SCHEMBL21362791 0.73 ALDH1A1 (0.44) ACHEALDH1A1NPSR1PTPN1PDF
SCHEMBL20158011 0.71 CA12 (0.38) ACHEBCHEALDH1A1MTNR1AMTNR1B
SCHEMBL20158055 0.70 CA12 (0.38) ACHEBCHEALDH1A1MTNR1AMTNR1B
SCHEMBL21362443 0.69 TAS2R14 (0.35) ACHEBCHEALDH1A1MTNR1AMTNR1B
SCHEMBL18393340 0.68 MAPT (0.44) PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed