SCHEMBL20159670

SCHEMBL20159670

C=C1C(N)C2CN(c3ccnc(Cl)c3)C12

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LOX P28300 1/20 0.32
LOXL3 P58215 1/20 0.32
LOXL2 Q9Y4K0 1/20 0.32
CYP17A1 P05093 4/20 0.32
CHRM4 P08173 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23504833 0.77 CHRM4 (0.37) LOXLOXL3LOXL2CYP17A1CHRM4
SCHEMBL20159731 0.76 MMP2 (0.31)
SCHEMBL20159356 0.72 CHRM4 (0.32) LOXLOXL3LOXL2CYP17A1CHRM4
SCHEMBL20159647 0.70 CHRNB2 (0.40) LOXLOXL3LOXL2CYP17A1
SCHEMBL20159656 0.66 CHRNA3 (0.39) LOXLOXL3LOXL2CYP17A1CHRM4
SCHEMBL20159609 0.66 CYP17A1 (0.38) LOXLOXL3LOXL2CYP17A1CHRM4
SCHEMBL18970901 0.65 CHRM4 (0.38) LOXLOXL3LOXL2CYP17A1CHRM4
SCHEMBL20609194 0.65 CHRM4 (0.38) LOXLOXL3LOXL2CYP17A1CHRM4
SCHEMBL20609193 0.65 CHRM4 (0.38) LOXLOXL3LOXL2CYP17A1CHRM4
SCHEMBL20031740 0.65 CHRM4 (0.38) LOXLOXL3LOXL2CYP17A1CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538516-B1 PHENOXYTRIAZOLES HOFFMANN LA ROCHE (CH) 2021-06-16 EP disclosed
WO-2018087018-A1 PHENOXYTRIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2018-05-17 WO disclosed