SCHEMBL20161336

SCHEMBL20161336

N=C(c1nc(F)n(Cc2ccccc2)n1)c1cccnc1NCc1ccccc1F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
ENPP2 Q13822 1/20 0.39
KDM4E B2RXH2 3/20 0.39
F2 P00734 1/20 0.37
F10 P00742 1/20 0.37
LMNA P02545 3/20 0.36
THRB P10828 1/20 0.36
AURKA O14965 1/20 0.36
RPS6KB1 P23443 1/20 0.36
SMN1; SMN2 Q16637 4/20 0.35
ABL1 P00519 2/20 0.35
SRC P12931 2/20 0.35
TP53 P04637 2/20 0.35
POLB P06746 2/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
HSD17B10 Q99714 1/20 0.35
GAA P10253 1/20 0.34
MEN1 O00255 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22874060 0.75 AURKA (0.43) KDM4ELMNAAURKARPS6KB1SMN1; SMN2
SCHEMBL20161096 0.70 STAT6 (0.47) ALDH1A1KDM4ESMN1; SMN2MAPK1GAA
SCHEMBL20161518 0.70 CASP6 (0.43) ALDH1A1KDM4ELMNAAURKARPS6KB1
SCHEMBL20161209 0.70 AURKA (0.40) ALDH1A1KDM4ELMNAAURKARPS6KB1
SCHEMBL19146434 0.70 LMNA (0.35) ALDH1A1KDM4ELMNAAURKARPS6KB1
SCHEMBL18359723 0.70 SLC26A6 (0.36) ALDH1A1KDM4ELMNAAURKARPS6KB1
SCHEMBL22213515 0.70 LMNA (0.38) ALDH1A1KDM4ELMNAAURKARPS6KB1
SCHEMBL19241027 0.70 RPS6KB1 (0.37) ALDH1A1KDM4ELMNAAURKARPS6KB1
SCHEMBL19240910 0.70 AURKA (0.37) ALDH1A1KDM4ELMNAAURKARPS6KB1
SCHEMBL20161113 0.69 RPS6KB1 (0.41) ALDH1A1KDM4ELMNAAURKARPS6KB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089330-A2 SGC STIMULATORS IRONWOOD PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed