SCHEMBL20161113

SCHEMBL20161113

N=C(c1n[nH]c(=O)[nH]1)c1cccnc1NCc1ccccc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 2/20 0.41
AURKA O14965 1/20 0.41
LMNA P02545 2/20 0.40
KDM4E B2RXH2 3/20 0.39
MAPT P10636 3/20 0.39
GAA P10253 1/20 0.39
EGFR P00533 1/20 0.37
VNN1 O95497 1/20 0.37
CDC7 O00311 2/20 0.36
PLK4 O00444 1/20 0.36
CHEK1 O14757 1/20 0.36
DAPK3 O43293 1/20 0.36
RPS6KA5 O75582 1/20 0.36
MAP4K4 O95819 1/20 0.36
CHEK2 O96017 1/20 0.36
PIM1 P11309 1/20 0.36
PRKACA P17612 1/20 0.36
AKT1 P31749 1/20 0.36
AKT2 P31751 1/20 0.36
FLT4 P35916 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20161518 0.83 CASP6 (0.43) RPS6KB1AURKALMNAKDM4EEGFR
SCHEMBL20161209 0.82 AURKA (0.40) RPS6KB1AURKALMNAKDM4EMAPT
SCHEMBL20149081 0.81 KDM4E (0.38) RPS6KB1AURKALMNAKDM4EGAA
SCHEMBL20161268 0.80 ACHE (0.36) RPS6KB1AURKALMNAKDM4ECASP6
SCHEMBL20161291 0.80 LMNA (0.39) RPS6KB1AURKALMNAKDM4EGAA
SCHEMBL20161118 0.77 CSNK1D (0.46) KDM4EMAPTGAAHTTALDH1A1
SCHEMBL20161301 0.77 SMN1; SMN2 (0.55) LMNAMEN1KMT2ANPC1HTT
SCHEMBL20161340 0.77 CYP11B1 (0.35) RPS6KB1AURKALMNAKDM4EMAPT
SCHEMBL20161335 0.74 KDM4E (0.37) RPS6KB1AURKALMNAKDM4EMAPT
SCHEMBL22874060 0.72 AURKA (0.43) RPS6KB1AURKALMNAKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089330-A2 SGC STIMULATORS IRONWOOD PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed