SCHEMBL20161209

SCHEMBL20161209

N=C(c1nc(N)n[nH]1)c1cccnc1NCc1ccccc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.40
RPS6KB1 P23443 1/20 0.40
KDM4E B2RXH2 2/20 0.39
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
LMNA P02545 2/20 0.37
MAPT P10636 1/20 0.37
HTT P42858 1/20 0.37
ALDH1A1 P00352 2/20 0.36
EGFR P00533 1/20 0.36
MAP4K4 O95819 1/20 0.36
NTRK1 P04629 1/20 0.35
NTRK3 Q16288 1/20 0.35
NTRK2 Q16620 1/20 0.35
ROCK1 Q13464 1/20 0.35
CASP6 P55212 3/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20161291 0.87 LMNA (0.39) AURKARPS6KB1KDM4EMEN1KMT2A
SCHEMBL20149081 0.86 KDM4E (0.38) AURKARPS6KB1KDM4EMEN1KMT2A
SCHEMBL20161113 0.82 RPS6KB1 (0.41) AURKARPS6KB1KDM4EMEN1KMT2A
SCHEMBL20161518 0.82 CASP6 (0.43) AURKARPS6KB1KDM4EMEN1KMT2A
SCHEMBL20161301 0.80 SMN1; SMN2 (0.55) MEN1KMT2ALMNAHTTNPC1
SCHEMBL20161118 0.80 CSNK1D (0.46) KDM4EMAPTHTTALDH1A1POLB
SCHEMBL20161268 0.80 ACHE (0.36) AURKARPS6KB1KDM4EMEN1KMT2A
SCHEMBL20161340 0.80 CYP11B1 (0.35) AURKARPS6KB1KDM4EMEN1KMT2A
SCHEMBL20161335 0.79 KDM4E (0.37) AURKARPS6KB1KDM4EMEN1KMT2A
SCHEMBL22874060 0.78 AURKA (0.43) AURKARPS6KB1KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089330-A2 SGC STIMULATORS IRONWOOD PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed