SCHEMBL20161518

SCHEMBL20161518

N=C(c1ncn[nH]1)c1cccnc1NCc1ccccc1F

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CASP6 P55212 5/20 0.43
AURKA O14965 2/20 0.42
RPS6KB1 P23443 2/20 0.42
KDM4E B2RXH2 2/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
LMNA P02545 1/20 0.39
ALDH1A1 P00352 2/20 0.38
EGFR P00533 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CDC7 O00311 1/20 0.36
CCNE1 P24864 1/20 0.36
CDK2 P24941 1/20 0.36
DBF4 Q9UBU7 1/20 0.36
VNN1 O95497 1/20 0.36
PDPK1 O15530 1/20 0.35
NTRK1 P04629 1/20 0.35
NTRK3 Q16288 1/20 0.35
NTRK2 Q16620 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20161113 0.83 RPS6KB1 (0.41) CASP6AURKARPS6KB1KDM4EMEN1
SCHEMBL20161209 0.82 AURKA (0.40) CASP6AURKARPS6KB1KDM4EMEN1
SCHEMBL20149081 0.80 KDM4E (0.38) CASP6AURKARPS6KB1KDM4EMEN1
SCHEMBL20161291 0.79 LMNA (0.39) CASP6AURKARPS6KB1KDM4EMEN1
SCHEMBL20161301 0.75 SMN1; SMN2 (0.55) MEN1KMT2ALMNASMN1; SMN2
SCHEMBL20161118 0.75 CSNK1D (0.46) KDM4EALDH1A1SMN1; SMN2CCNE1CDK2
SCHEMBL20161268 0.74 ACHE (0.36) CASP6AURKARPS6KB1KDM4EMEN1
SCHEMBL20161340 0.74 CYP11B1 (0.35) AURKARPS6KB1KDM4EMEN1KMT2A
SCHEMBL22874060 0.74 AURKA (0.43) CASP6AURKARPS6KB1KDM4EMEN1
SCHEMBL20161335 0.74 KDM4E (0.37) AURKARPS6KB1KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089330-A2 SGC STIMULATORS IRONWOOD PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed