SCHEMBL20170624

SCHEMBL20170624

COc1ccc2c3c1O[C@@H]1C(OC(C)=O)=CCC(CC2)C31

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 7/20 0.35
MTNR1B P49286 7/20 0.35
NQO2 P16083 2/20 0.35
GABRA1 P14867 2/20 0.33
GABRB2 P47870 2/20 0.33
POLB P06746 1/20 0.32
NR3C1 P04150 1/20 0.32
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
HTR1A P08908 1/20 0.31
DRD2 P14416 2/20 0.31
DRD1 P21728 2/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
HSD17B10 Q99714 1/20 0.31
ABCB1 P08183 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20170617 0.88 HTR1A (0.32) MTNR1AMTNR1BNQO2HTR1A
SCHEMBL20170676 0.88 HTR1A (0.32) MTNR1AMTNR1BNQO2HTR1A
SCHEMBL20170600 0.76 OPRM1 (0.39) MTNR1AMTNR1BNQO2KDM4ELMNA
SCHEMBL20170645 0.76 OPRM1 (0.39) MTNR1AMTNR1BNQO2KDM4ELMNA
SCHEMBL20170640 0.73 HTR1A (0.34) HTR1ADRD2
SCHEMBL20170697 0.73 HTR1A (0.34) HTR1ADRD2
SCHEMBL20170753 0.73 GABRA1 (0.39) MTNR1AMTNR1BNQO2GABRA1GABRB2
SCHEMBL20170592 0.71 MTNR1A (0.40) MTNR1AMTNR1BNQO2POLBKDM4E
SCHEMBL20170728 0.68 OPRM1 (0.37) MTNR1AMTNR1BNQO2
SCHEMBL20170607 0.68 OPRM1 (0.37) MTNR1AMTNR1BNQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2453895-B1 (+) - MORPHINANS AS ANTAGONISTS OF TOLL-LIKE RECEPTOR 9 AND THERAPEUTIC USES THEREOF MALLINCKRODT LLC (US) 2018-05-23 EP disclosed