SCHEMBL20189708

SCHEMBL20189708

NC(=O)CCC(Nc1ccc2ccccc2c1)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.51
MMP2 P08253 2/20 0.47
MMP9 P14780 2/20 0.47
CYP1A2 P05177 2/20 0.47
RAB9A P51151 3/20 0.44
MAPT P10636 2/20 0.44
NPC1 O15118 2/20 0.44
MEN1 O00255 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
POLB P06746 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
GAA P10253 2/20 0.43
ALDH1A1 P00352 2/20 0.42
CYP3A4 P08684 1/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
SLC1A3 P43003 1/20 0.42
SLC1A2 P43004 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20189709 1.00 KMT2A (0.51) KMT2AMMP2MMP9CYP1A2RAB9A
SCHEMBL27076462 0.87 SLC1A3 (0.48) MMP2MMP9SLC1A3SLC1A2SLC1A1
SCHEMBL7274405 0.84 GGH (0.52) KMT2AMMP9CYP1A2RAB9AMAPT
SCHEMBL7274402 0.84 GGH (0.52) KMT2AMMP9CYP1A2RAB9AMAPT
SCHEMBL27657427 0.84 RAB9A (0.47) KMT2ACYP1A2RAB9AMAPTNPC1
SCHEMBL3448329 0.84 KMT2A (0.64) KMT2AMMP2MMP9MAPTL3MBTL1
SCHEMBL3448327 0.84 KMT2A (0.64) KMT2AMMP2MMP9MAPTL3MBTL1
SCHEMBL2820711 0.83 PPARG (0.54) KMT2ACYP1A2RAB9AMAPTNPC1
SCHEMBL27469903 0.83 PPARG (0.54) KMT2ACYP1A2RAB9AMAPTNPC1
Hydrochloric Acid SCHEMBL23834278 0.82 KMT2A (0.62) KMT2AMMP2MMP9MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 123 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250353814-A1 NON-PEPTIDIC CELL-PENETRATING MOTIFS OHIO STATE INNOVATION FOUNDATION (US) 2025-11-20 US claimed
US-12404236-B2 Non-peptidic cell-penetrating motifs OHIO STATE INNOVATION FOUNDATION (US) 2025-09-02 US claimed
US-12329799-B2 Peptidyl inhibitors of calcineurin-NFAT interaction OHIO STATE INNOVATION FOUNDATION (US) 2025-06-17 US claimed
US-20240101509-A1 NON-PEPTIDIC CELL-PENETRATING MOTIFS OHIO STATE INNOVATION FOUNDATION 2024-03-28 US claimed
CN-117567639-A Polypeptide conjugates for intracellular delivery of binding peptides 俄亥俄州国家创新基金会 2024-02-20 CN claimed
US-20240033318-A1 PEPTIDYL INHIBITORS OF CALCINEURIN-NFAT INTERACTION OHIO STATE INNOVATION FOUNDATION 2024-02-01 US claimed
US-11814341-B2 Non-peptidic cell-penetrating motifs OHIO STATE INNOVATION FOUNDATION (US) 2023-11-14 US claimed
US-20230212235-A1 LOOPED PROTEINS COMPRISING CELL PENETRATING PEPTIDES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-07-06 US claimed
CN-115135665-A Cyclic proteins comprising cell penetrating peptides 俄亥俄州国家创新基金会 2022-09-30 CN claimed
WO-2021138397-A1 LOOPED PROTEINS COMPRISING CELL PENETRATING PEPTIDES OHIO STATE INNOVATION FOUNDATION (US) 2021-07-08 WO claimed
US-20260125426-A1 CYCLIC CELL-PENETRATING PEPTIDES AND USES THEREOF OHIO STATE INNOVATION FOUNDATION (US) 2026-05-07 US disclosed
US-20260098262-A9 COMPOUNDS AND METHODS FOR SKIPPING EXON 44 IN DUCHENNE MUSCULAR DYSTROPHY ENTRADA THERAPEUTICS INC (US) 2026-04-09 US disclosed
US-20260070947-A1 CYCLIC CELL-PENETRATING PEPTIDE COMPOUNDS OHIO STATE INNOVATION FOUNDATION (US) 2026-03-12 US disclosed
US-20260070948-A1 CYCLIC CELL-PENETRATING PEPTIDES WITH CARGO OHIO STATE INNOVATION FOUNDATION (US) 2026-03-12 US disclosed
EP-4706689-A2 COMPOSITIONS FOR DELIVERY OF ANTISENSE COMPOUNDS Entrada Therapeutics, Inc. (US) 2026-03-11 EP disclosed
EP-3544623-A1 CELL-PENETRATING PEPTIDE SEQUENCES Ohio State Innovation Foundation (US) 2019-10-02 EP disclosed
WO-2019148194-A2 PEPTIDYL INHIBITORS OF CALCINEURIN-NFAT INTERACTION OHIO STATE INNOVATION FOUNDATION (US) 2019-08-01 WO disclosed
WO-2019148195-A2 CYCLIC PEPTIDYL INHIBITORS OF CAL-PDZ BINDING DOMAIN OHIO STATE INNOVATION FOUNDATION (US) 2019-08-01 WO disclosed
WO-2019070962-A1 BICYCLIC PEPTIDYL INHIBITORS OHIO STATE INNOVATION FOUNDATION (US) 2019-04-11 WO disclosed
WO-2018098231-A1 CELL-PENETRATING PEPTIDE SEQUENCES OHIO STATE INNOVATION FOUNDATION (US) 2018-05-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12404236-B2 Non-peptidic cell-penetrating motifs TIMM50, TIMM10, PITRM1 KMT2A 4862/4885MMP2 1219/4885MMP9 2041/4885
US-20240101509-A1 NON-PEPTIDIC CELL-PENETRATING MOTIFS TIMM50, TIMM10, PITRM1 KMT2A 4862/4885MMP2 1219/4885MMP9 2041/4885
US-20250353814-A1 NON-PEPTIDIC CELL-PENETRATING MOTIFS TIMM50, TIMM10, PITRM1 KMT2A 4862/4885MMP2 1219/4885MMP9 2041/4885
US-20230212235-A1 LOOPED PROTEINS COMPRISING CELL PENETRATING PEPTIDES LNPEP, SPPL2B, CNBP KMT2A 4379/4885MMP2 629/4885MMP9 1192/4885
US-20260098262-A9 COMPOUNDS AND METHODS FOR SKIPPING EXON 44 IN DUCHENNE MUSCULAR DYSTROPHY UTRN, SMN1; SMN2, UPF1 KMT2A 2310/4885MMP2 3212/4885MMP9 2724/4885
US-20260125426-A1 CYCLIC CELL-PENETRATING PEPTIDES AND USES THEREOF SLC7A1, TAP1, SLC7A5 KMT2A 2819/4885MMP2 1466/4885MMP9 702/4885
US-20260070947-A1 CYCLIC CELL-PENETRATING PEPTIDE COMPOUNDS SLC7A1, SLC38A7, SLC6A19 KMT2A 4374/4885MMP2 339/4885MMP9 355/4885
US-11814341-B2 Non-peptidic cell-penetrating motifs TIMM50, TIMM10, PITRM1 KMT2A 4862/4885MMP2 1219/4885MMP9 2041/4885
US-20260070948-A1 CYCLIC CELL-PENETRATING PEPTIDES WITH CARGO SLC7A1, SLC38A7, SLC6A19 KMT2A 3978/4885MMP2 550/4885MMP9 734/4885
US-12329799-B2 Peptidyl inhibitors of calcineurin-NFAT interaction CHP1, NFATC1, PPP3R1 KMT2A 3612/4885MMP2 3863/4885MMP9 4113/4885
US-20240033318-A1 PEPTIDYL INHIBITORS OF CALCINEURIN-NFAT INTERACTION CHP1, NFATC1, PPP3R1 KMT2A 3612/4885MMP2 3863/4885MMP9 4113/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.