SCHEMBL20195282

SCHEMBL20195282

BC(B)(B)C(B)(B)Oc1ccc(CCO)cn1

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 1/20 0.33
CA2 P00918 1/20 0.33
CYP4F2 P78329 3/20 0.32
CYP4A11 Q02928 3/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
ALOX5 P09917 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
BACE1 P56817 1/20 0.31
HRH3 Q9Y5N1 2/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20195208 0.84 PPARA (0.40) PPARACA2CYP4F2CYP4A11KDM4E
SCHEMBL20195263 0.79 L3MBTL1 (0.36) PPARACA2CYP4F2CYP4A11KDM4E
SCHEMBL20195262 0.75 CA2 (0.32) CA2
SCHEMBL3229511 0.74 NNMT (0.44) CYP4F2CYP4A11KDM4EMAPT
SCHEMBL20195249 0.73 MAPT (0.50) CA2CYP4F2CYP4A11KDM4EALDH1A1
SCHEMBL30942648 0.73 CA2 (0.38) CA2CYP4F2CYP4A11KDM4EALDH1A1
SCHEMBL9388917 0.72 L3MBTL1 (0.54) MAPT
SCHEMBL23309376 0.72 PPARA (0.44) PPARACYP4F2CYP4A11
SCHEMBL22558607 0.71 PPARA (0.38) PPARACA2CYP4F2CYP4A11KDM4E
SCHEMBL18402496 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2729447-B1 POSITIVE ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTOR H LUNDBECK AS (DK) 2018-05-30 EP disclosed