SCHEMBL20195263

SCHEMBL20195263

BC(B)(B)COc1ccc(CCO)cn1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.36
CA2 P00918 1/20 0.34
CYP4F2 P78329 4/20 0.34
CYP4A11 Q02928 4/20 0.34
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
ALOX5 P09917 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
BACE1 P56817 1/20 0.32
FFAR1 O14842 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
PPARA Q07869 2/20 0.31
PPARG P37231 1/20 0.31
CD274 Q9NZQ7 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
PIK3CD O00329 1/20 0.30
PIK3CA P42336 1/20 0.30
PIK3CB P42338 1/20 0.30
PI4KA P42356 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9388917 0.83 L3MBTL1 (0.54) L3MBTL1MAPT
SCHEMBL20195282 0.79 PPARA (0.33) CA2CYP4F2CYP4A11KDM4EALDH1A1
SCHEMBL20195208 0.79 PPARA (0.40) CA2CYP4F2CYP4A11KDM4EALDH1A1
SCHEMBL30942648 0.77 CA2 (0.38) L3MBTL1CA2CYP4F2CYP4A11KDM4E
SCHEMBL20195249 0.77 MAPT (0.50) L3MBTL1CA2CYP4F2CYP4A11KDM4E
SCHEMBL20195262 0.76 CA2 (0.32) CA2
SCHEMBL3229511 0.75 NNMT (0.44) CYP4F2CYP4A11KDM4EMAPTPIK3CA
SCHEMBL23309220 0.75 DGAT1 (0.55) L3MBTL1CYP4F2CYP4A11PPARA
SCHEMBL20195254 0.75 ACACB (0.42) L3MBTL1CYP4F2CYP4A11KDM4EALDH1A1
SCHEMBL22558708 0.74 L3MBTL1 (0.51) L3MBTL1CYP4F2CYP4A11MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2729447-B1 POSITIVE ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTOR H LUNDBECK AS (DK) 2018-05-30 EP disclosed