SCHEMBL20195208

SCHEMBL20195208

BC(B)(C)Oc1ccc(CCO)cn1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 6/20 0.40
CYP4F2 P78329 7/20 0.36
CYP4A11 Q02928 7/20 0.36
CA2 P00918 1/20 0.33
PPARG P37231 4/20 0.33
CDK1 P06493 1/20 0.33
KDR P35968 1/20 0.33
FFAR1 O14842 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
ALOX5 P09917 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
BACE1 P56817 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20195282 0.84 PPARA (0.33) PPARACYP4F2CYP4A11CA2KDM4E
SCHEMBL20195263 0.79 L3MBTL1 (0.36) PPARACYP4F2CYP4A11CA2PPARG
SCHEMBL23309376 0.78 PPARA (0.44) PPARACYP4F2CYP4A11PPARG
SCHEMBL3229511 0.78 NNMT (0.44) CYP4F2CYP4A11KDM4EMAPT
SCHEMBL20195249 0.76 MAPT (0.50) CYP4F2CYP4A11CA2FFAR1KDM4E
SCHEMBL20195262 0.75 CA2 (0.32) CA2
SCHEMBL20195254 0.73 ACACB (0.42) PPARACYP4F2CYP4A11PPARGKDM4E
SCHEMBL20195258 0.73 ACACB (0.47) CYP4F2CYP4A11ALDH1A1
SCHEMBL2938892 0.73 PPARG (0.39) PPARACYP4F2CYP4A11PPARGKDM4E
SCHEMBL30942648 0.73 CA2 (0.38) CYP4F2CYP4A11CA2FFAR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2729447-B1 POSITIVE ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTOR H LUNDBECK AS (DK) 2018-05-30 EP disclosed