SCHEMBL20197243

SCHEMBL20197243

FC(F)(F)SNc1ccc(-c2csc(-c3ccnc4[nH]ccc34)n2)c(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 4/20 0.45
CIT O14578 3/20 0.40
RHEB Q15382 2/20 0.39
ABL1 P00519 1/20 0.38
BCR P11274 1/20 0.38
ROCK1 Q13464 4/20 0.38
PRKCI P41743 2/20 0.37
AXL P30530 1/20 0.37
CCNK O75909 2/20 0.35
CDK12 Q9NYV4 2/20 0.35
BRAF P15056 1/20 0.35
IKBKB O14920 1/20 0.34
CHUK O15111 1/20 0.34
DAPK3 O43293 1/20 0.34
JAK2 O60674 1/20 0.34
PRKD3 O94806 1/20 0.34
MAP4K4 O95819 1/20 0.34
PAK4 O96013 1/20 0.34
CSF1R P07333 1/20 0.34
RET P07949 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20197303 0.86 CYP1A2 (0.32) NUDT1RPS6KA3
SCHEMBL20197271 0.84 MEN1 (0.39) RHEBABL1BCRKDRCYP19A1
SCHEMBL16535266 0.83 NUDT1 (0.43) NUDT1CITRHEBABL1BCR
SCHEMBL20197336 0.80 CYP19A1 (0.46) CYP19A1
SCHEMBL20197228 0.79 CYP1A1 (0.42) CYP19A1
SCHEMBL20197355 0.78 MEN1 (0.53)
SCHEMBL20197440 0.78 KDM4E (0.36) CYP19A1
SCHEMBL20197249 0.78 SREBF2 (0.43)
SCHEMBL20197221 0.78 SREBF2 (0.55)
SCHEMBL20197302 0.78 SMN1; SMN2 (0.46) CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3038622-B1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECH LLC (US) 2018-05-30 EP disclosed