SCHEMBL20197303

SCHEMBL20197303

Fc1cnc2[nH]ccc2c1-c1nc(-c2ccc(NSC(F)(F)F)cc2Cl)cs1

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.32
CYP1B1 Q16678 4/20 0.32
CYP1A1 P04798 2/20 0.32
TGFBR1 P36897 2/20 0.32
CYP2C8 P10632 1/20 0.32
NUDT1 P36639 1/20 0.31
RPS6KA3 P51812 1/20 0.31
AMY1A P0DUB6 1/20 0.31
KDM4E B2RXH2 1/20 0.30
NPC1 O15118 1/20 0.30
CRHBP P24387 1/20 0.30
RAB9A P51151 1/20 0.30
CRHR2 Q13324 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20197243 0.86 NUDT1 (0.45) NUDT1RPS6KA3
SCHEMBL16535520 0.84 PTGS1 (0.35) CYP1A2CYP1B1CYP1A1TGFBR1KDM4E
SCHEMBL20197271 0.81 MEN1 (0.39) CYP1A2CYP1B1CYP1A1KDM4ENPC1
SCHEMBL20197228 0.76 CYP1A1 (0.42) CYP1A2CYP1B1CYP1A1AMY1AKDM4E
SCHEMBL20197355 0.75 MEN1 (0.53) KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL20197302 0.74 SMN1; SMN2 (0.46) CYP1A2CYP1B1CYP1A1KDM4ENPC1
SCHEMBL20197318 0.74 EIF4E (0.46) CYP1A2CYP1B1CYP1A1AMY1AKDM4E
SCHEMBL20197342 0.73 LMNA (0.37) CYP1A2CYP1B1CYP1A1AMY1AKDM4E
SCHEMBL20197336 0.72 CYP19A1 (0.46) CYP1A2CYP1B1CYP1A1AMY1AKDM4E
SCHEMBL20197220 0.72 SREBF2 (0.35) AMY1AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3038622-B1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECH LLC (US) 2018-05-30 EP disclosed