Bromide

Bromide

SCHEMBL20202

Br.CCCCC(CNC(=O)c1ccc(C(C)CO)c([N+](=O)[O-])c1)C(P)(CCCC)CCCC

nearest known ligand 0.38

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 7/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 7/20 0.37
GAA P10253 4/20 0.37
MAPK1 P28482 3/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ALDH1A1 P00352 7/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HTT P42858 2/20 0.36
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HPGD P15428 2/20 0.35
ATM Q13315 1/20 0.35
HSP90AA1 P07900 1/20 0.35
HCAR3 P49019 2/20 0.35
PDK1 Q15118 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL20203 0.78 LMNA (0.48) LMNAPOLBMAPTGAAMEN1
Bromide SCHEMBL12474014 0.76 ALDH1A1 (0.47) LMNAPOLBMAPTGAAMEN1
SCHEMBL25650 0.74 LMNA (0.51) LMNAPOLBMAPTGAAMEN1
SCHEMBL16016907 0.71 THRA (0.48) MAPTGAAALDH1A1HCAR3PDK1
SCHEMBL16016753 0.69 ESR1 (0.55) LMNAPOLBMAPTMAPK1KMT2A
SCHEMBL21319 0.69 CASP6 (0.57) LMNAMEN1KMT2ATSHRHCAR3
SCHEMBL2949996 0.68 VCAM1 (0.54) LMNAPOLBMAPTMEN1KMT2A
SCHEMBL16016735 0.66 THRA (0.41) MAPTGAAHCAR3PDK1
SCHEMBL2947165 0.66 PDK1 (0.46) LMNAPOLBMAPTKMT2AALDH1A1
SCHEMBL29887339 0.66 PDK1 (0.46) LMNAPOLBMAPTKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2748176-A1 IONIC TAGS FOR SYNTHESIS OF OLIGORIBONUCLEOTIDES The Royal Institution for the Advancement of Learning / McGill University (CA) 2014-07-02 EP disclosed
WO-2013026142-A1 IONIC TAGS FOR SYNTHESIS OF OLIGORIBONUCLEOTIDES THE ROYAL INSTITUTION FOR THE ADVANCEMENT OF LEARNING/MCGILL UNIVERSITY (CA) 2013-02-28 WO disclosed