SCHEMBL20204633

SCHEMBL20204633

CCC(F)COc1cccc(CCNCc2cnc(CN3CC(=S)NC3=O)cn2)c1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 8/20 0.35
BCHE P06276 2/20 0.34
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
DUT P33316 2/20 0.33
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ALDH1A1 P00352 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
ADRB2 P07550 2/20 0.32
ADRB1 P08588 2/20 0.32
DRD3 P35462 1/20 0.32
ADRB3 P13945 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20204885 0.85 BCHE (0.36) BCHENOS3NOS1NOS2KDM4E
SCHEMBL20204886 0.85 MCHR1 (0.35) BCHENOS3NOS1NOS2KDM4E
SCHEMBL20204636 0.74 CXCR4 (0.36) BCHEDUTMEN1KMT2AALDH1A1
SCHEMBL21536566 0.67 DUT (0.45) DUTKDM4EALDH1A1
SCHEMBL20204894 0.62 BCHE (0.40) CYP2D6BCHENOS3NOS1NOS2
SCHEMBL21536718 0.62 DUT (0.43) DUTALDH1A1
SCHEMBL21536596 0.60 DUT (0.43) DUTALDH1A1
SCHEMBL5223504 0.60 BCHE (0.66) CYP2D6BCHEKDM4EALDH1A1
SCHEMBL27586255 0.59 HSD17B10 (0.52) KDM4EMEN1KMT2ATDP1HCRTR1
SCHEMBL18183457 0.59 MTNR1A (0.58)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018098209-A1 AMINO SULFONYL COMPOUNDS CV6 THERAPEUTICS (NI) LIMITED (GB) 2018-05-31 WO disclosed