SCHEMBL202301

SCHEMBL202301

CC(C)(C)OC(=O)N1CSCC1C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.48
ATM Q13315 1/20 0.47
HSD17B10 Q99714 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.38
USP2 O75604 1/20 0.38
PREP P48147 2/20 0.37
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
RECQL P46063 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1022969 1.00 ACE (0.48) ACEATMHSD17B10SMN1; SMN2USP2
SCHEMBL202300 1.00 ACE (0.48) ACEATMHSD17B10SMN1; SMN2USP2
SCHEMBL16187224 0.87 ATM (0.45) ACEATMHSD17B10SMN1; SMN2USP2
SCHEMBL14237836 0.87 ATM (0.45) ACEATMHSD17B10SMN1; SMN2USP2
SCHEMBL26077743 0.87 ATM (0.45) ACEATMHSD17B10SMN1; SMN2USP2
SCHEMBL1249539 0.87 HSD17B10 (0.46) ATMHSD17B10SMN1; SMN2USP2PREP
SCHEMBL3509553 0.85 ATM (0.44) ACEATMHSD17B10SMN1; SMN2USP2
SCHEMBL9879848 0.85 ATM (0.44) ACEATMHSD17B10SMN1; SMN2USP2
SCHEMBL3509552 0.85 ATM (0.44) ACEATMHSD17B10SMN1; SMN2USP2
SCHEMBL1021093 0.85 ATM (0.44) ACEATMHSD17B10SMN1; SMN2USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 180 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101090631-A Novel compounds for treatment of cancer and disorders associated with angiogenesis function UNIV SOUTHERN CALIFORNIA (US) 2007-12-19 CN claimed
US-20060142294-A1 Novel compounds for treatment of cancer and disorders associated with angiogenesis function UNIVERSITY OF SOUTHERN CALIFORNIA 2006-06-29 US claimed
US-20250368637-A1 SOLID-STATE FORMS OF N-(2-(4-CYANOTHIAZOLIDIN-3-YL)-2-OXOETHYL)-6-MORPHOLINOQUINOLINE-4-CARBOXAMIDE ASTRAZENECA AB (SE) 2025-12-04 US disclosed
US-12415835-B2 Peptide-compound cyclization method CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2025-09-16 US disclosed
US-20250170104-A1 INHIBITORS OF PSEUDOMONAS AERUGINOSA VIRULENCE FACTOR Lasß HELMHOLTZ ZENTRUM INFEKTIONSFORSCHUNG GMBH (DE) 2025-05-29 US disclosed
EP-4486452-A1 INHIBITORS OF PSEUDOMONAS AERUGINOSA VIRULENCE FACTOR LASSS Helmholtz-Zentrum für Infektionsforschung GmbH (DE) 2025-01-08 EP disclosed
WO-2024215870-A2 HETEROCYCLIC COMPOUNDS AS INHIBITORS OF POLYMERASE THETA AND METHODS OF USE THEREOF 1CBIO, INC. (US) 2024-10-17 WO disclosed
US-20240166689-A1 PEPTIDE-COMPOUND CYCLIZATION METHOD CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2024-05-23 US disclosed
US-20240101549-A1 N-(2-(4-CYANOTHIAZOLIDIN-3-YL)-2-OXOETHYL)-QUINOLINE-4-CARBOXAMIDES ASTRAZENECA AB (SE) 2024-03-28 US disclosed
US-11891457-B2 Peptide-compound cyclization method CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2024-02-06 US disclosed
US-11858924-B2 N-(2-(4-cyanothiazolidin-3-yl)-2-oxoethyl)-quinoline-4-carboxamides ASTRAZENECA (SE) 2024-01-02 US disclosed
WO-1992014732-A1 INDOLES USEFUL AS PLATELET ACTIVATING FACTOR ANTAGONISTS ABBOTT LABORATORIES (US) 1992-09-03 WO disclosed
EP-0490667-A2 HIV protease inhibitors JAPAN ENERGY CORPORATION (JP) 1992-06-17 EP disclosed
WO-1992001668-A1 BENZOIC ACID SUBSTITUTED DERIVATIVES HAVING CARDIOVASCULAR ACTIVITY ITALFARMACO S.P.A. (IT) 1992-02-06 WO disclosed
EP-0213326-B1 2,5-DIMETHYL PYRROLE DERIVATIVES, THEIR PREPARATION AND THEIR USE CASSELLA Aktiengesellschaft (DE) 1991-03-06 EP disclosed
EP-0388909-A2 Thiazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1990-09-26 EP disclosed
EP-0175363-B1 4,5-DIHYDRO-3(2H)-PYRIDAZINONES, PROCESS FOR THEIR PREPARATION AND THEIR USE CASSELLA Aktiengesellschaft (DE) 1990-01-17 EP disclosed
US-4837225-A ENCEPHALOTROPIC AND PSYCHOTROPIC EFFECTS CASSELL AKTIENGESELLSCHAFT (DE) 1989-06-06 US disclosed
US-4816454-A CARDIOVASCULAR DISORDERS CASSELLA AKTIENGESELLSCHAFT (DE) 1989-03-28 US disclosed
EP-0213326-A1 2,5-Dimethyl pyrrole derivatives, their preparation and their use CASSELLA Aktiengesellschaft (DE) 1987-03-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11891457-B2 Peptide-compound cyclization method VIP, NGLY1, GLP1R ACE 621/4885ATM 3913/4885HSD17B10 3115/4885
US-20060142294-A1 Novel compounds for treatment of cancer and disorders associated with angiogenesis function VEGFA, TEK, LIPG ACE 4837/4885ATM 1955/4885HSD17B10 2660/4885
US-20240166689-A1 PEPTIDE-COMPOUND CYCLIZATION METHOD VIP, NGLY1, GLP1R ACE 621/4885ATM 3913/4885HSD17B10 3115/4885
US-20250170104-A1 INHIBITORS OF PSEUDOMONAS AERUGINOSA VIRULENCE FACTOR Lasß LTA, SERPINB1, LAS1L ACE 606/4885ATM 3938/4885HSD17B10 1790/4885
US-20250368637-A1 SOLID-STATE FORMS OF N-(2-(4-CYANOTHIAZOLIDIN-3-YL)-2-OXOETHYL)-6-MORPHOLINOQUINOLINE-4-CARBOXAMIDE FAP, FIBP, DNPEP ACE 50/4885ATM 3109/4885HSD17B10 4631/4885
US-20240101549-A1 N-(2-(4-CYANOTHIAZOLIDIN-3-YL)-2-OXOETHYL)-QUINOLINE-4-CARBOXAMIDES FAP, PREP, CTRL ACE 30/4885ATM 4050/4885HSD17B10 4763/4885
US-12415835-B2 Peptide-compound cyclization method VIP, NGLY1, GLP1R ACE 621/4885ATM 3913/4885HSD17B10 3115/4885
US-11858924-B2 N-(2-(4-cyanothiazolidin-3-yl)-2-oxoethyl)-quinoline-4-carboxamides FAP, PREP, CTRL ACE 30/4885ATM 4050/4885HSD17B10 4763/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.