SCHEMBL20239299

SCHEMBL20239299

CNS(=O)(=O)Cc1ccc(Oc2cc(CN)ccn2)cc1

nearest known ligand 0.57

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 20/20 0.57
LOX P28300 17/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18249838 0.84 LOXL2 (0.62) LOXL2LOX
SCHEMBL20239304 0.82 LOXL2 (0.43) LOXL2LOX
SCHEMBL20239300 0.81 LOXL2 (0.42) LOXL2LOX
SCHEMBL18249748 0.81 P2RX3 (0.47) LOXL2
SCHEMBL18249869 0.81 KDM4E (0.40) LOXL2LOX
SCHEMBL20239160 0.80 PGR (0.37) LOXL2LOX
SCHEMBL20239198 0.80 DGAT2 (0.37) LOXL2LOX
SCHEMBL20239324 0.80 VNN1 (0.41) LOXL2LOX
SCHEMBL20472862 0.79 LOXL2 (0.58) LOXL2LOX
SCHEMBL20239285 0.78 VNN1 (0.38) LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3298001-B1 DGAT2 INHIBITORS LILLY CO ELI (US) 2020-05-13 EP disclosed
US-10053429-B2 DGAT2 inhibitors ELI LILLY AND COMPANY (US) 2018-08-21 US disclosed
US-20180162825-A1 NOVEL DGAT2 INHIBITORS ELI LILY AND COMPANY (US) 2018-06-14 US disclosed
US-20180162825-A1 NOVEL DGAT2 INHIBITORS ELI LILY AND COMPANY (US) 2018-06-14 US disclosed
US-20180162825-A1 NOVEL DGAT2 INHIBITORS ELI LILY AND COMPANY (US) 2018-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180162825-A1 NOVEL DGAT2 INHIBITORS DGAT2, DGAT1, LCAT LOXL2 2081/4885LOX 2453/4885
US-10053429-B2 DGAT2 inhibitors DGAT2, DGAT1, LCAT LOXL2 1951/4885LOX 2250/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.