SCHEMBL20274140

SCHEMBL20274140

O=C(CO)N1CCN(Cc2oc3ccc(Cl)cc3c2Cl)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.48
TSHR P16473 2/20 0.48
KDM4E B2RXH2 1/20 0.48
POLB P06746 3/20 0.45
KMT2A Q03164 1/20 0.44
AKR1C3 P42330 2/20 0.42
HTR2A P28223 1/20 0.42
HTR2B P41595 1/20 0.42
EPHX2 P34913 1/20 0.41
CYP3A4 P08684 2/20 0.40
LMNA P02545 2/20 0.40
ABCB11 O95342 1/20 0.40
CYP1A2 P05177 1/20 0.40
ADRA2A P08913 1/20 0.40
CYP2D6 P10635 1/20 0.40
CHRM1 P11229 1/20 0.40
TBXA2R P21731 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20274136 0.88 MEN1 (0.42) TSHRKMT2ACYP2D6CYP2C19
SCHEMBL20274170 0.85 L3MBTL1 (0.44) ALDH1A1KDM4EKMT2ALMNATBXAS1
SCHEMBL20274139 0.77 HRH4 (0.47) ALDH1A1TSHRKDM4EPOLBKMT2A
SCHEMBL20274205 0.75 SOS1 (0.51) KMT2AAKR1C3EPHX2LMNAKCNH2
SCHEMBL20274216 0.75 HTR2B (0.46) ALDH1A1TSHRKDM4EPOLBKMT2A
SCHEMBL20274189 0.72 L3MBTL1 (0.44) ALDH1A1KDM4EPOLBKMT2ATBXAS1
SCHEMBL20274113 0.71 SIGMAR1 (0.39) ALDH1A1TSHRKDM4EKMT2AAKR1C3
SCHEMBL20274204 0.70 EPHX2 (0.40) ALDH1A1TSHRKDM4EPOLBKMT2A
SCHEMBL20274196 0.69 HRH4 (0.73) ALDH1A1KDM4ELMNAHSD17B10
SCHEMBL2958198 0.66 MAPT (0.50) ALDH1A1TSHRKDM4EPOLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3428162-B1 ANTHELMINTIC COMPOUNDS AND COMPOSITIONS AND METHOD OF USING THEREOF BOEHRINGER INGELHEIM ANIMAL HEALTH USA INC (US) 2021-05-05 EP disclosed
EP-2922845-B1 ANTHELMINTIC COMPOUNDS AND COMPOSITIONS AND METHOD OF USING THEREOF MERIAL INC (US) 2018-06-20 EP disclosed