SCHEMBL20340469

SCHEMBL20340469

COc1cc(N2C(=O)NC(=O)C23CCCCC3)ccn1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 3/20 0.37
QPCT Q16769 1/20 0.36
IDH1 O75874 1/20 0.36
MAT2A P31153 1/20 0.36
ELOVL1 Q9BW60 1/20 0.35
ALDH1A1 P00352 1/20 0.34
MAPK1 P28482 1/20 0.34
EGLN1 Q9GZT9 3/20 0.34
PTH1R Q03431 1/20 0.34
POLB P06746 1/20 0.33
LOX P28300 1/20 0.33
LOXL2 Q9Y4K0 1/20 0.33
CHRNA7 P36544 1/20 0.33
RPS6KA2 Q15349 1/20 0.32
SLC6A9 P48067 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL721033 0.81 CHRNB2 (0.44) IDH1ALDH1A1MAPK1
SCHEMBL20340466 0.80 CYP17A1 (0.38) CYP17A1IDH1MAT2AELOVL1ALDH1A1
SCHEMBL190640 0.75 ALDH1A1 (0.55) ALDH1A1MAPK1POLB
SCHEMBL201840 0.73 POLB (0.51) ALDH1A1MAPK1POLBSLC6A9
SCHEMBL18961831 0.70 LMNA (0.46) SLC6A9
SCHEMBL719564 0.69 CYP11B1 (0.45) CHRNA7SLC6A9
SCHEMBL2544529 0.68 MMP13 (0.46) QPCTSLC6A9
SCHEMBL17077228 0.67 MAPT (0.45) ALDH1A1SLC6A9
SCHEMBL421867 0.67 AKR1B1 (0.37) QPCTALDH1A1MAPK1POLBSLC6A9
SCHEMBL242118 0.67 SLC6A3 (0.40) QPCT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10011601-B2 Substituted spirocyclic inhibitors of autotaxin X-RX, INC. (US) 2018-07-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10011601-B2 Substituted spirocyclic inhibitors of autotaxin ENPP2, SLC10A1, CXCR3 CYP17A1 230/4885QPCT 550/4885IDH1 2459/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.