SCHEMBL14944729

SCHEMBL14944729

CC(C)(C)c1c[nH]c(-c2nc(N)c3c(n2)N(Cc2ccccc2)CN3)n1

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.32
ADORA3 P0DMS8 1/20 0.31
ADORA2A P29274 1/20 0.31
TLR7 Q9NYK1 1/20 0.30
THRB P10828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14944653 0.82 DRD2 (0.31) ALDH1A1ADORA3ADORA2A
SCHEMBL14944658 0.80 TLR7 (0.36) ALDH1A1ADORA3ADORA2ATLR7THRB
SCHEMBL14944685 0.76 TLR7 (0.33) TLR7
SCHEMBL14944688 0.75 ALDH1A1 (0.30) ALDH1A1
SCHEMBL19423858 0.75 CCR5 (0.31) ALDH1A1TLR7THRB
SCHEMBL20343752 0.74 ADORA2A (0.39) ADORA3ADORA2ATLR7
SCHEMBL28852897 0.72 HSP90AA1 (0.40) ALDH1A1TLR7THRB
SCHEMBL16206184 0.71 TLR7 (0.59) TLR7
SCHEMBL14944686 0.69 TLR7 (0.33) TLR7
SCHEMBL20343748 0.69 GSK3A (0.43) ALDH1A1TLR7THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9556176-B2 Purine derivatives for the treatment of viral infections JANSSEN SCIENCES IRELAND UC (IE) 2017-01-31 US disclosed
WO-2013068438-A1 PURINE DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS JANSSEN R&D IRELAND (IE) 2013-05-16 WO disclosed