SCHEMBL14944658

SCHEMBL14944658

Cc1nc(-c2nc(N)c3c(n2)N(Cc2ccccc2)CN3)[nH]c1C

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 5/20 0.36
ADORA3 P0DMS8 2/20 0.32
ADORA2A P29274 2/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
THRB P10828 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
NPY5R Q15761 1/20 0.31
TYMS P04818 1/20 0.31
ADORA1 P30542 1/20 0.31
POLB P06746 2/20 0.30
GAA P10253 1/20 0.30
RGS12 O14924 1/20 0.30
USP2 O75604 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14944685 0.87 TLR7 (0.33) TLR7
SCHEMBL14944729 0.80 ALDH1A1 (0.32) TLR7ADORA3ADORA2AALDH1A1THRB
SCHEMBL19423858 0.79 CCR5 (0.31) TLR7ALDH1A1THRB
SCHEMBL20343752 0.76 ADORA2A (0.39) TLR7ADORA3ADORA2AMAPK1ADORA1
SCHEMBL14944653 0.76 DRD2 (0.31) ADORA3ADORA2AALDH1A1MAPK1MAPT
SCHEMBL28852897 0.75 HSP90AA1 (0.40) TLR7KDM4EALDH1A1THRBTSHR
SCHEMBL14944688 0.72 ALDH1A1 (0.30) ALDH1A1
SCHEMBL20343756 0.69 TLR7 (0.41) TLR7ALDH1A1MEN1KMT2A
SCHEMBL4144591 0.69 HPRT1 (0.50) TYMS
SCHEMBL14944686 0.66 TLR7 (0.33) TLR7ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068438-A1 PURINE DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS JANSSEN R&D IRELAND (IE) 2013-05-16 WO disclosed